SCHEMBL8364653

SCHEMBL8364653

CC(C)Oc1cccc(C(C(=O)N(C)CCCCO)c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ACHE P22303 3/20 0.38
BCHE P06276 2/20 0.38
FAAH O00519 1/20 0.38
TACR1 P25103 2/20 0.37
SLC6A9 P48067 1/20 0.37
ATM Q13315 1/20 0.36
SLC6A2 P23975 4/20 0.35
SLC6A4 P31645 4/20 0.35
SLC6A3 Q01959 4/20 0.35
CYP3A4 P08684 4/20 0.35
CYP2D6 P10635 4/20 0.35
OPRK1 P41145 1/20 0.35
CYP1A2 P05177 1/20 0.35
TSHR P16473 1/20 0.35
THPO P40225 1/20 0.35
MARK4 Q96L34 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8366249 0.86 ALDH1A1 (0.39) KDM4EALDH1A1LMNASMN1; SMN2ACHE
SCHEMBL8365000 0.81 SLC6A3 (0.39) KDM4EALDH1A1LMNASMN1; SMN2TACR1
SCHEMBL8124968 0.72 TACR1 (0.36) ALDH1A1LMNASMN1; SMN2TACR1SLC6A9
SCHEMBL8970550 0.69 TACR1 (0.42) TACR1CYP3A4CYP2D6OPRK1CYP1A2
Hydrochloric Acid SCHEMBL8430668 0.69 TACR2 (0.39) TACR1SLC6A2SLC6A4SLC6A3
SCHEMBL8364651 0.69 CCR5 (0.46) TACR1
SCHEMBL7599760 0.69 KDM4E (0.63) KDM4ELMNATACR1ATMCYP2D6
SCHEMBL8366286 0.68 MEN1 (0.47) ALDH1A1SMN1; SMN2TACR1SLC6A2SLC6A4
SCHEMBL8561473 0.67 TACR1 (0.42) TACR1CYP3A4CYP2D6OPRK1CYP1A2
SCHEMBL8369232 0.67 MEN1 (0.46) ALDH1A1SMN1; SMN2TACR1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939411-A PIPERIDINE DERIVATIVES SUBSTITUTED AT POSITION 4 WITH NEW FUNCTIONS OTHER THAN THOSE DESCRIBED PREVIOUSLY HAVE A HIGH AFFINITY FOR NEUROKININ RECEPTORS AND ARE USEFUL FOR TREATMENT OF SUBSTANCE P AND NEUROKININ DEPENDENT PATHOLOGIES SANOFI (FR) 1999-08-17 US disclosed
US-5830906-A Piperidine derivatives, process for obtaining them and pharmaceutical compositions containing them SANOFI (FR) 1998-11-03 US disclosed