SCHEMBL8366343

SCHEMBL8366343

COc1cc(O)cc(OS(=O)(=O)c2cccc3c(N(C)C)cccc23)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.49
F2 P00734 3/20 0.48
PRSS1 P07477 3/20 0.48
PRSS2 P07478 3/20 0.48
PRSS3 P35030 3/20 0.48
EDNRA P25101 8/20 0.47
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
HTT P42858 1/20 0.45
HIF1A Q16665 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
TYMS P04818 2/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43
KDM4E B2RXH2 1/20 0.42
NSD2 O96028 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL711797 0.80 CA2 (0.58) CA2F2PRSS1PRSS2PRSS3
SCHEMBL16610066 0.77 TYMS (0.53) CA2F2PRSS1PRSS2PRSS3
SCHEMBL12603022 0.76 CA2 (0.65) CA2F2PRSS1PRSS2PRSS3
SCHEMBL6750357 0.76 F2 (0.59) F2HTTTDP1L3MBTL1KMT2A
SCHEMBL8366342 0.75 F2 (0.42) CA2F2PRSS2EDNRACYP1A2
SCHEMBL714171 0.75 CA2 (0.52) CA2F2PRSS1PRSS2PRSS3
SCHEMBL18487536 0.75 KDM4E (0.48) CA2F2PRSS1PRSS2PRSS3
SCHEMBL7440192 0.73 F2 (0.55) F2PRSS2KMT2AKDM4EHSD17B10
SCHEMBL714494 0.72 TYMS (0.57) CA2F2PRSS1PRSS2PRSS3
SCHEMBL18487742 0.72 DYRK1A (0.41) CA2F2PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883405-A4 AMIDINO PROTEASE INHIBITORS DIMENSIONAL PHARM INC (US) 1999-04-28 EP disclosed
EP-0883405-A1 AMIDINO PROTEASE INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 1998-12-16 EP disclosed
WO-1997024135-A1 AMIDINO PROTEASE INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 1997-07-10 WO disclosed