SCHEMBL8366356

SCHEMBL8366356

COc1ccc2[nH]c(=O)cc(CCO)c2c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.63
KDM4E B2RXH2 7/20 0.58
ALDH1A1 P00352 6/20 0.58
L3MBTL1 Q9Y468 2/20 0.58
GAA P10253 2/20 0.58
POLB P06746 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
KMT2A Q03164 3/20 0.51
MEN1 O00255 2/20 0.51
HSD17B10 Q99714 2/20 0.51
MAPT P10636 2/20 0.51
TSHR P16473 2/20 0.51
GFER P55789 1/20 0.51
HPGD P15428 4/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
ABCG2 Q9UNQ0 1/20 0.48
GPR84 Q9NQS5 1/20 0.47
GHSR Q92847 1/20 0.46
MTNR1A P48039 1/20 0.46
AKR1C2 P52895 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8364405 0.86 KDM4E (0.55) CYP2D6KDM4EALDH1A1L3MBTL1GAA
SCHEMBL8366255 0.82 KDM4E (0.67) KDM4EALDH1A1L3MBTL1GAAPOLB
SCHEMBL9152213 0.81 ALDH1A1 (0.48) KDM4EALDH1A1L3MBTL1GAAPOLB
SCHEMBL8369457 0.81 KDM4E (0.59) CYP2D6KDM4EALDH1A1L3MBTL1GAA
SCHEMBL29375720 0.78 CYP2D6 (1.00) CYP2D6KDM4EALDH1A1L3MBTL1TDP1
SCHEMBL676574 0.78 CYP2D6 (1.00) CYP2D6KDM4EALDH1A1L3MBTL1TDP1
SCHEMBL2267796 0.77 ALDH1A1 (0.66) KDM4EALDH1A1L3MBTL1GAAPOLB
SCHEMBL9160413 0.77 KDM4E (0.46) KDM4EALDH1A1GAAKMT2AMEN1
SCHEMBL2798566 0.77 KDM4E (0.75) KDM4EALDH1A1L3MBTL1GAAPOLB
Hydrochloric Acid SCHEMBL9293745 0.76 KDM4E (0.56) KDM4EALDH1A1L3MBTL1GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850235-B1 QUINOLEIN-2(1H)-ONE DERIVATIVES AS SEROTONIN ANTAGONISTS SANOFI SYNTHELABO (FR) 1999-12-01 EP disclosed
US-5958924-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS, RESTENOSIS, ANTICOALUGANTS, RESPIRATORY SYSTEM DISORDERS SYNTHELABO (FR) 1999-09-28 US disclosed
EP-0850235-A1 QUINOLEIN-2(1H)-ONE DERIVATIVES AS SEROTONIN ANTAGONISTS SYNTHELABO (FR) 1998-07-01 EP disclosed
WO-1997010238-A1 QUINOLEIN-2(1H)-ONE DERIVATIVES AS SEROTONIN ANTAGONISTS SYNTHELABO (FR) 1997-03-20 WO disclosed