SCHEMBL8366372

SCHEMBL8366372

COC(=O)Cc1cc(=O)n(C)c2ccc(OC)cc12

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
KDM4E B2RXH2 1/20 0.56
HPGD P15428 1/20 0.56
AKR1C3 P42330 6/20 0.54
MTNR1A P48039 4/20 0.47
MTNR1B P49286 4/20 0.47
NQO2 P16083 2/20 0.47
AKR1C2 P52895 2/20 0.46
PKM P14618 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CNR2 P34972 1/20 0.45
PTGS2 P35354 1/20 0.45
RXFP1 Q9HBX9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8366206 0.88 KDM4E (0.55) ALDH1A1KDM4EHPGDAKR1C3AKR1C2
SCHEMBL8366324 0.84 THRB (0.47) ALDH1A1KDM4EHPGDPOLBMAPT
SCHEMBL8367855 0.84 HPGD (0.43) ALDH1A1KDM4EHPGDAKR1C3POLB
SCHEMBL9152250 0.82 MAPT (0.59) ALDH1A1KDM4EHPGDNQO2POLB
SCHEMBL2686296 0.81 MTNR1A (0.65) AKR1C3MTNR1AMTNR1BNQO2AKR1C2
SCHEMBL8367875 0.81 BRD4 (0.45) ALDH1A1KDM4EHPGDAKR1C3AKR1C2
SCHEMBL8648192 0.77 AKR1C3 (0.68) ALDH1A1AKR1C3MTNR1AMTNR1BNQO2
SCHEMBL6208739 0.76 MAPT (0.56) ALDH1A1KDM4EHPGDMTNR1AMTNR1B
SCHEMBL8369457 0.75 KDM4E (0.59) ALDH1A1KDM4EHPGDAKR1C3MTNR1A
SCHEMBL29187763 0.74 AKR1C3 (0.47) ALDH1A1KDM4EHPGDAKR1C3MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958924-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS, RESTENOSIS, ANTICOALUGANTS, RESPIRATORY SYSTEM DISORDERS SYNTHELABO (FR) 1999-09-28 US disclosed