SCHEMBL8368908

SCHEMBL8368908

Cc1ccc(S(=O)(=O)ON2CCC(NC(=O)NC3CCCC3)(c3ccccc3)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.47
ALDH1A1 P00352 5/20 0.45
POLB P06746 2/20 0.45
TP53 P04637 1/20 0.45
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 1/20 0.42
EPHX2 P34913 1/20 0.42
FPR1 P21462 2/20 0.41
USP2 O75604 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 2/20 0.40
NPC1 O15118 1/20 0.40
EPHX1 P07099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744607 0.84 POLB (0.57) ALDH1A1POLBMEN1KMT2AHPGD
SCHEMBL8367979 0.84 HTT (0.47) ALDH1A1POLBCNR1CNR2MEN1
SCHEMBL8368924 0.84 ENPP3 (0.46) ALDH1A1POLBMEN1KMT2ALMNA
SCHEMBL6447443 0.83 POLB (0.45) ALDH1A1POLBMEN1KMT2ALMNA
SCHEMBL7750046 0.83 POLB (0.45) ALDH1A1POLBMEN1KMT2ARAB9A
SCHEMBL8368905 0.83 KMT2A (0.43) ALDH1A1POLBMEN1KMT2AUSP2
SCHEMBL7679125 0.82 POLB (0.43) ALDH1A1POLBMEN1KMT2ASMN1; SMN2
SCHEMBL8368906 0.81 ADORA3 (0.47) ADORA3ALDH1A1POLBTP53CNR1
SCHEMBL7678500 0.80 POLB (0.47) ALDH1A1POLBMEN1KMT2ASMN1; SMN2
SCHEMBL6470098 0.79 POLB (0.46) ALDH1A1POLBMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965580-A TREATMENT OF SUBSTANCE P- AND NEUROKININ-DEPENDENT DISORDERS SANOFI (FR) 1999-10-12 US disclosed
US-5939411-A PIPERIDINE DERIVATIVES SUBSTITUTED AT POSITION 4 WITH NEW FUNCTIONS OTHER THAN THOSE DESCRIBED PREVIOUSLY HAVE A HIGH AFFINITY FOR NEUROKININ RECEPTORS AND ARE USEFUL FOR TREATMENT OF SUBSTANCE P AND NEUROKININ DEPENDENT PATHOLOGIES SANOFI (FR) 1999-08-17 US disclosed
US-5830906-A Piperidine derivatives, process for obtaining them and pharmaceutical compositions containing them SANOFI (FR) 1998-11-03 US disclosed