SCHEMBL8375006

SCHEMBL8375006

COC(=O)NCCOc1cc(-c2ccccc2)on1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.46
TP53 P04637 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CYP1A2 P05177 2/20 0.46
HPGD P15428 2/20 0.46
NPC1 O15118 1/20 0.46
CYP2C19 P33261 1/20 0.46
HIF1A Q16665 2/20 0.46
POLB P06746 1/20 0.46
FAAH O00519 2/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 1/20 0.44
KMT2A Q03164 1/20 0.44
STAT3 P40763 1/20 0.44
STAT1 P42224 1/20 0.44
CHRM4 P08173 2/20 0.43
CHRM5 P08912 2/20 0.43
CHRM1 P11229 2/20 0.43
CHRM3 P20309 2/20 0.43
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8375785 0.89 MTNR1A (0.54) RAB9ATP53SMN1; SMN2CYP1A2HPGD
SCHEMBL8378941 0.88 GABRA5 (0.46) RAB9ASMN1; SMN2HIF1AFAAHMAPK1
SCHEMBL8375557 0.86 BCHE (0.47) FAAHHDAC3HDAC1HDAC2HDAC10
SCHEMBL8380154 0.85 SMN1; SMN2 (0.55) RAB9ATP53SMN1; SMN2CYP1A2HPGD
Hydrochloric Acid SCHEMBL8378876 0.83 CHRM4 (0.46) RAB9ASMN1; SMN2NPC1ALDH1A1CHRM4
SCHEMBL8378917 0.81 BCHE (0.49) HDAC3HDAC1HDAC2HDAC10HDAC8
SCHEMBL8380141 0.78 NPC1 (0.51) RAB9ATP53SMN1; SMN2CYP1A2HPGD
SCHEMBL8375005 0.78 RAB9A (0.59) RAB9ATP53SMN1; SMN2CYP1A2HPGD
SCHEMBL8375021 0.78 BCHE (0.57)
SCHEMBL8375551 0.78 HDAC1 (0.44) RAB9ASMN1; SMN2NPC1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
CN-1216986-A Isoxazole derivatives SANKYO CO (JP) 1999-05-19 CN disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed