SCHEMBL8375135

SCHEMBL8375135

CCN(CC)C(=O)Oc1cnccc1N

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 2/20 0.44
KDM4E B2RXH2 4/20 0.44
LMNA P02545 5/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TSHR P16473 1/20 0.43
ALDH1A1 P00352 2/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
P2RX4 Q99571 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7364409 0.83 MEN1 (0.50) MEN1KMT2AHSD17B10KDM4ELMNA
SCHEMBL8375858 0.83 KDM4E (0.46) MEN1KMT2AKDM4ELMNAL3MBTL1
SCHEMBL7368604 0.82 LMNA (0.54) MEN1KMT2AHSD17B10KDM4ELMNA
SCHEMBL8375863 0.81 MEN1 (0.47) MEN1KMT2AHSD17B10KDM4ELMNA
SCHEMBL29956916 0.81 LMNA (0.49) MEN1KMT2AHSD17B10KDM4ELMNA
SCHEMBL8376699 0.79 MEN1 (0.46) MEN1KMT2AHSD17B10KDM4ELMNA
SCHEMBL14566738 0.79 ALDH1A1 (0.51) MEN1KMT2AHSD17B10KDM4ELMNA
SCHEMBL8376712 0.78 HSD17B10 (0.66) MEN1KMT2AHSD17B10KDM4ELMNA
SCHEMBL4634558 0.78 KDM4E (0.51) MEN1KMT2AHSD17B10KDM4EL3MBTL1
SCHEMBL8375140 0.77 KDM6B (0.51) MEN1KMT2AHSD17B10KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821239-A USEFUL FOR TREATING ALZHEIMER'S DISEASE CAUSED BY CHOLINERGIC DEFICIT FROMMER LAWRENCE & HUAG LLP (US) 1998-10-13 US claimed
US-5869480-A ALLEVIATING MEMORY DYSFUNCTION CHARACTERIZED BY CHOLINERGIC DEFICIT HOECHST MARION ROUSSEL INC. (US) 1999-02-09 US disclosed
US-5866565-A ALZHEIMER'S DISORDERS HOECHST MARION ROUSSEL INC. (US) 1999-02-02 US disclosed
US-5821239-A USEFUL FOR TREATING ALZHEIMER'S DISEASE CAUSED BY CHOLINERGIC DEFICIT FROMMER LAWRENCE & HUAG LLP (US) 1998-10-13 US disclosed
EP-0477903-B1 Substituted-4-amino-3-pyridinols, a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-04-03 EP disclosed
EP-0477903-A2 Substituted-4-amino-3-pyridinols, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-04-01 EP disclosed