SCHEMBL8375534

SCHEMBL8375534

c1ccc(-c2cc(OCCN3CCCCC3)no2)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.55
CHRM4 P08173 1/20 0.55
CHRM5 P08912 1/20 0.55
CHRM3 P20309 1/20 0.55
HRH3 Q9Y5N1 4/20 0.55
CXCR1 P25024 1/20 0.55
BACE1 P56817 1/20 0.54
PTPN1 P18031 2/20 0.53
LTA4H P09960 2/20 0.52
CHRM2 P08172 1/20 0.52
DRD1 P21728 1/20 0.52
SLC6A2 P23975 1/20 0.52
ADRA1A P35348 1/20 0.52
OPRM1 P35372 1/20 0.52
DRD3 P35462 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8375520 0.99 CHRM1 (0.54) CHRM1CHRM4CHRM5CHRM3HRH3
SCHEMBL8379062 0.99 CHRM1 (0.56) CHRM1CHRM4CHRM5CHRM3HRH3
Hydrochloric Acid SCHEMBL8380152 0.97 CHRM1 (0.55) CHRM1CHRM4CHRM5CHRM3HRH3
SCHEMBL8380069 0.88 NPC1 (0.56) HRH3CXCR1PTPN1LTA4HDRD1
Hydrochloric Acid SCHEMBL8380005 0.87 NPC1 (0.59) HRH3PTPN1LTA4H
Hydrochloric Acid SCHEMBL8377507 0.86 LTA4H (0.47) CHRM1CHRM4CHRM5CHRM3CXCR1
SCHEMBL21121342 0.82 CXCR1 (0.79) HRH3CXCR1PTPN1LTA4H
SCHEMBL21121935 0.82 CXCR1 (0.79) HRH3CXCR1PTPN1LTA4H
SCHEMBL8376242 0.78 SCD5 (0.52) CHRM1CHRM4CHRM5CHRM3CXCR1
SCHEMBL5617855 0.76 RAB9A (0.47) CHRM1CHRM4CHRM5CHRM3CXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed