SCHEMBL8375559

SCHEMBL8375559

CC(C)(C)ON(C=O)CCOc1cc(-c2ccc(-c3ccccc3)cc2)on1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR1 P25024 2/20 0.41
CHRM4 P08173 2/20 0.39
CHRM5 P08912 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMPD1 P17405 1/20 0.35
CASP3 P42574 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PTGS2 P35354 1/20 0.34
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8378946 0.98 CXCR1 (0.40) CXCR1CHRM4CHRM5CHRM1CHRM3
SCHEMBL8378925 0.92 CXCR1 (0.41) CXCR1NPC1RAB9A
SCHEMBL8375555 0.90 NPC1 (0.35) CXCR1NPC1RAB9ACASP3SENP8
SCHEMBL8379540 0.89 ALDH1A1 (0.38) CXCR1CHRM4CHRM5CHRM1CHRM3
SCHEMBL8375770 0.89 CXCR1 (0.43) CXCR1NPC1RAB9ASMPD1
SCHEMBL8376906 0.89 CXCR1 (0.40) CXCR1NPC1RAB9APTGS2
SCHEMBL8378889 0.89 CXCR1 (0.32) CXCR1CHRM4CHRM5CHRM1CHRM3
SCHEMBL8375023 0.89 SMPD1 (0.47) CXCR1SMPD1
SCHEMBL8380142 0.88 HPGD (0.42) CXCR1NPC1RAB9AALDH1A1
SCHEMBL8375816 0.88 EPHX2 (0.38) CXCR1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed