SCHEMBL8377409

SCHEMBL8377409

CC(C)c1c(OCCNC(=O)OC(C)(C)C)noc1-c1ccccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.41
ALDH1A1 P00352 3/20 0.41
MALT1 Q9UDY8 1/20 0.40
LMNA P02545 3/20 0.40
TSHR P16473 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SCN9A Q15858 1/20 0.39
KCNA5 P22460 1/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
HPGD P15428 2/20 0.38
GAA P10253 1/20 0.38
IDO1 P14902 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
PPARD Q03181 1/20 0.37
STK17B O94768 1/20 0.37
STK17A Q9UEE5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8377390 0.89 IDO1 (0.46) PDK2ALDH1A1MEN1KMT2ACA12
SCHEMBL8375760 0.86 IDO1 (0.43) PDK2ALDH1A1MALT1MEN1KMT2A
SCHEMBL8376442 0.84 LMNA (0.40) ALDH1A1LMNATSHRMEN1KMT2A
SCHEMBL8375676 0.83 RAB9A (0.41) PDK2MALT1LMNATSHRKMT2A
SCHEMBL8375796 0.82 ADORA2A (0.43) ALDH1A1TSHRSCN9ACA12CA1
SCHEMBL8377351 0.81 CA12 (0.40) PDK2SCN9ACA12CA1CA2
SCHEMBL8377384 0.81 SCN9A (0.41) PDK2SCN9ACA12CA1CA2
SCHEMBL8378805 0.80 IDO1 (0.42) ALDH1A1LMNASCN9ACA12CA1
SCHEMBL8377356 0.79 S1PR1 (0.44) PDK2MALT1MEN1KMT2ASCN9A
SCHEMBL8380070 0.79 IDO1 (0.45) PDK2ALDH1A1LMNATSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed