SCHEMBL8377605

SCHEMBL8377605

CCCCCCC=CC(=O)N(C)Cc1ccc(O)c(OC)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.67
TRPV1 Q8NER1 5/20 0.65
CYP1A2 P05177 3/20 0.65
CYP3A4 P08684 3/20 0.65
CYP2D6 P10635 2/20 0.65
LTA4H P09960 2/20 0.65
CYP2C8 P10632 2/20 0.65
CYP2C9 P11712 2/20 0.65
CYP2B6 P20813 2/20 0.65
CYP2C19 P33261 2/20 0.65
CYP2E1 P05181 1/20 0.65
ALOX5 P09917 1/20 0.65
CYP2A6 P11509 1/20 0.65
MAPT P10636 2/20 0.58
HPGD P15428 2/20 0.58
MEN1 O00255 1/20 0.58
TP53 P04637 1/20 0.58
MTOR P42345 1/20 0.58
KMT2A Q03164 1/20 0.58
ALDH1A1 P00352 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16715940 0.86 TRPV1 (0.66) HTR1ATRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL27885589 0.82 HTR1A (0.70) HTR1ATRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL8622173 0.82 HTR1A (0.60) HTR1ATRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL4886657 0.81 HTR1A (1.00) HTR1ATRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL29564502 0.81 HTR1A (1.00) HTR1ATRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL4886648 0.81 HTR1A (1.00) HTR1ATRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL29929375 0.81 HTR1A (1.00) HTR1ATRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL4885163 0.81 HTR1A (1.00) HTR1ATRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL4885150 0.81 HTR1A (1.00) HTR1ATRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL30335074 0.81 HTR1A (1.00) HTR1ATRPV1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5985860-A System for transdermal delivery of pain relieving substances TOPPO, ROBERT J. 1999-11-16 US disclosed
US-5318960-A System for transdermal delivery of pain relieving substances Toppo, Frank (US) 1994-06-07 US disclosed