SCHEMBL8378902

SCHEMBL8378902

CC(C)(C)OC(=O)N[C@@H](Cc1ccc(-c2ccccc2C(=O)OC(C)(C)C)cc1)C(=O)OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.54
CTSS P25774 5/20 0.53
CTSK P43235 4/20 0.53
CTSB P07858 2/20 0.50
CTSL P07711 1/20 0.50
BCL2 P10415 1/20 0.49
PPARA Q07869 2/20 0.49
ACE P12821 1/20 0.48
KLK5 Q9Y337 1/20 0.48
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
POLB P06746 1/20 0.47
MAPK1 P28482 1/20 0.47
SRC P12931 1/20 0.46
PPARG P37231 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8379883 0.89 PTPN1 (0.61) PTPN1CTSSCTSKCTSBCTSL
SCHEMBL7409389 0.88 CTSS (0.65) PTPN1CTSSCTSKCTSBCTSL
SCHEMBL7409385 0.88 CTSS (0.65) PTPN1CTSSCTSKCTSBCTSL
SCHEMBL22404737 0.86 CTSS (0.64) CTSSCTSKCTSBCTSLPPARA
SCHEMBL85543 0.86 CTSS (0.64) CTSSCTSKCTSBCTSLPPARA
SCHEMBL3355326 0.86 CTSS (0.64) CTSSCTSKCTSBCTSLPPARA
SCHEMBL23729806 0.85 CTSS (0.58) PTPN1CTSSCTSKCTSBCTSL
SCHEMBL3826349 0.84 CTSS (0.66) PTPN1CTSSCTSKCTSBCTSL
SCHEMBL7235877 0.84 CTSS (0.63) CTSSCTSKCTSBCTSLPPARA
SCHEMBL1486267 0.84 CTSS (0.63) CTSSCTSKCTSBCTSLPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901628-A1 PHOSPHOTYROSINE MIMICS AND METHODS FOR IDENTIFYING AND USING SAME BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1999-03-17 EP disclosed
WO-1997042501-A1 PHOSPHOTYROSINE MIMICS AND METHODS FOR IDENTIFYING AND USING SAME BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1997-11-13 WO disclosed