SCHEMBL8380288

SCHEMBL8380288

C/C=C/CC1CCC(c2cnc(-c3ccc(F)c(Cl)c3)nc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNB3 Q05901 1/20 0.35
AXL P30530 1/20 0.35
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
MDM2 Q00987 2/20 0.34
DGAT1 O75907 2/20 0.33
TGFBR1 P36897 2/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
SLC9A1 P19634 3/20 0.33
GRM2 Q14416 1/20 0.33
KCNH2 Q12809 2/20 0.32
ACACB O00763 1/20 0.32
DHODH Q02127 1/20 0.32
NISCH Q9Y2I1 1/20 0.32
TGFBR2 P37173 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8383726 0.91 CYP11B1 (0.34) S1PR1S1PR3DGAT1CYP11B1CYP11B2
SCHEMBL8380302 0.90 ACACB (0.36) CYP11B1CYP11B2GRM2ACACBDHODH
SCHEMBL8381991 0.90 S1PR3 (0.36) S1PR1S1PR3DGAT1CYP11B1CYP11B2
SCHEMBL8517281 0.86 GRM2 (0.35) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL8382675 0.86 HDAC4 (0.35) S1PR1S1PR3DGAT1
SCHEMBL8383609 0.82 S1PR1 (0.36) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL8383601 0.82 S1PR1 (0.36) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL9312273 0.82 S1PR1 (0.36) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL9312474 0.80 CHRNB1 (0.35) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL8380287 0.80 CHRNB1 (0.35) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0475273-B1 Liquid crystal mixture containing halogenated alcenyl compounds MERCK PATENT GMBH (DE) 1999-04-07 EP disclosed
EP-0475273-A1 Halogenated alcenyl compounds F. HOFFMANN-LA ROCHE AG (CH) 1992-03-18 EP disclosed