SCHEMBL8380302

SCHEMBL8380302

C/C=C/CC1CCC(c2cnc(-c3ccc(F)c(F)c3)nc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.36
NPY5R Q15761 1/20 0.35
GRIN2B Q13224 5/20 0.34
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32
PDE5A O76074 1/20 0.31
CYP11B2 P19099 2/20 0.31
HDAC4 P56524 1/20 0.31
CYP17A1 P05093 1/20 0.31
CYP3A4 P08684 1/20 0.31
GRM2 Q14416 1/20 0.31
OPRL1 P41146 1/20 0.31
KDM1A O60341 1/20 0.30
CYP11B1 P15538 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
GAA P10253 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
CACNA1H O95180 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8383726 0.90 CYP11B1 (0.34) ACACBGRIN2BCYP11B2CYP11B1CYP1A2
SCHEMBL8380288 0.90 CHRNB1 (0.35) ACACBCYP11B2GRM2CYP11B1DHODH
SCHEMBL8380281 0.87 KDM1A (0.40) GRIN2BCYP11B2GRM2KDM1ACYP11B1
SCHEMBL8517670 0.85 NPY5R (0.34) ACACBNPY5RGRIN2BPDGFRBPDGFRA
SCHEMBL8380306 0.85 CYP3A4 (0.33) NPY5RGRIN2BCYP11B2CYP17A1CYP3A4
SCHEMBL8382675 0.84 HDAC4 (0.35) HDAC4KDM1A
SCHEMBL8381991 0.83 S1PR3 (0.36) PDGFRBPDGFRACYP11B2HDAC4CYP11B1
SCHEMBL9247689 0.82 CHRNB2 (0.34) NPY5RGRIN2BPDGFRBPDGFRAGRM2
SCHEMBL8378335 0.81 PDGFRB (0.33) ACACBGRIN2BPDGFRBPDGFRAPDE5A
SCHEMBL8378334 0.81 PDGFRB (0.33) ACACBGRIN2BPDGFRBPDGFRAPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0475273-B1 Liquid crystal mixture containing halogenated alcenyl compounds MERCK PATENT GMBH (DE) 1999-04-07 EP disclosed
EP-0475273-A1 Halogenated alcenyl compounds F. HOFFMANN-LA ROCHE AG (CH) 1992-03-18 EP disclosed