SCHEMBL8380458

SCHEMBL8380458

COCCOc1c(Cl)c([CH]C(=O)OC(c2ccccc2)c2ccccc2)c(OC)c(Cl)c1OCCOC

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
HPGD P15428 3/20 0.33
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
TNFRSF1A P19438 1/20 0.32
KMT2A Q03164 1/20 0.31
APEX1 P27695 1/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
LMNA P02545 2/20 0.31
MAPT P10636 1/20 0.31
SLC6A5 Q9Y345 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
KDM4E B2RXH2 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
PDE4D Q08499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8381669 0.93 ALDH1A1 (0.34) ALDH1A1HPGDHTR1AADRA1DADRA1A
SCHEMBL8381851 0.92 ALDH1A1 (0.33) ALDH1A1HPGDHTR1AADRA1DADRA1A
SCHEMBL8381832 0.83 ALDH1A1 (0.36) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8378617 0.82 MAPK1 (0.35) ALDH1A1HPGDHTR1AADRA1DADRA1A
SCHEMBL8381498 0.82 ALDH1A1 (0.39) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8377870 0.81 MAPK1 (0.33) ALDH1A1HPGDHTR1AADRA1DADRA1A
SCHEMBL8379003 0.81 ALDH1A1 (0.36) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8381714 0.76 LMNA (0.39) ALDH1A1HPGDHTR1AADRA1DADRA1A
SCHEMBL8679133 0.76 ALDH1A1 (0.34) ALDH1A1HPGDHTR1AADRA1DADRA1A
SCHEMBL8382692 0.74 HTR1A (0.35) ALDH1A1HPGDHTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883248-A QUATERNARY AMMONIUM INTERMEDIATES ROUSSEL UCLAF (FR) 1999-03-16 US disclosed
US-5763617-A Cephalosporins ROUSSEL UCLAF (FR) 1998-06-09 US disclosed
US-5728828-A A 3-(3-CHLORO- OR IODOPROP-1-EN-1-YL),7-(2-AMINOTHIAZOL-4-YL) ((CARBOXY)(PHENYL)METHOXYIMINO)ACETAMIDO-3-CEPHEM; GRAMNEGATIVE AND -POSITIVE BACTERIA, ESP. ANTIBIOTIC-RESISTANCE STAPHYLOCOCCUS ROUSSEL UCLAF (FR) 1998-03-17 US disclosed
US-5712266-A Cephalosporins ROUSSEL UCLAF (FR) 1998-01-27 US disclosed