SCHEMBL8382616

SCHEMBL8382616

CN1CC=C(c2ccc(O)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
QDPR P09417 3/20 1.00
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369176 0.84 QDPR (0.72) QDPR
SCHEMBL7744453 0.82 QDPR (1.00) QDPR
Hydrochloric Acid SCHEMBL10354108 0.81 QDPR (0.68) QDPRDRD2DRD4DRD3
SCHEMBL6043136 0.81 QDPR (0.68) QDPR
SCHEMBL578138 0.81 QDPR (0.68) QDPR
SCHEMBL1814323 0.81 QDPR (0.68) QDPR
SCHEMBL155267 0.81 QDPR (0.68) QDPR
SCHEMBL13898494 0.81 QDPR (0.68) QDPR
SCHEMBL16862164 0.80 QDPR (0.67) QDPR
SCHEMBL50923 0.80 QDPR (0.67) QDPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7425563-B2 Excellent poly (ADP-ribose) synthetase inhibitors; various ischemic diseases, inflammatory diseases, neurodegenerative diseases, diabetes, septic shock, cephalic injury; 1,2-Dihydro-4-[4-(dimethylaminomethyl)phenyl]-5-hydroxy-1-oxoisoquinoline KYORIN PHARMACEUTICAL CO., LTD. (JP) 2008-09-16 US disclosed
US-7425563-B2 Excellent poly (ADP-ribose) synthetase inhibitors; various ischemic diseases, inflammatory diseases, neurodegenerative diseases, diabetes, septic shock, cephalic injury; 1,2-Dihydro-4-[4-(dimethylaminomethyl)phenyl]-5-hydroxy-1-oxoisoquinoline KYORIN PHARMACEUTICAL CO., LTD. (JP) 2008-09-16 US disclosed
US-5874433-A Blocking utilization of tetrahydrobiopterin to block induction of nitric oxide synthesis CORNELL RESEARCH FOUNDATION, INC. (US) 1999-02-23 US disclosed
US-5502050-A DIHYDROXYPHENYL-SUBSTITITED PYRIDINES OR QUINONES, HYPERTENSIVE AGENTS CORNELL RESEARCH FOUNDATION, INC. (US) 1996-03-26 US disclosed