SCHEMBL8386348

SCHEMBL8386348

C[Si](C)(C)OC=Cc1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 8/20 0.48
TRPA1 O75762 3/20 0.44
NQO2 P16083 1/20 0.44
PTGS1 P23219 2/20 0.44
APP P05067 1/20 0.44
HSD11B1 P28845 1/20 0.41
ALOX5 P09917 1/20 0.40
PTGS2 P35354 1/20 0.40
FBP1 P09467 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8488639 0.79 AHR (0.43) NFE2L2PTGS1ALOX5PTGS2FBP1
SCHEMBL12495291 0.79 PTGS1 (0.42) NFE2L2NQO2PTGS1PTGS2
SCHEMBL770392 0.78 MAOB (0.44) NFE2L2TRPA1
SCHEMBL8491011 0.77 NPC1 (0.48) NFE2L2ALOX5
SCHEMBL9718330 0.76 NFE2L2 (0.59) NFE2L2TRPA1NQO2PTGS1APP
SCHEMBL10567248 0.75 NFE2L2 (0.54) NFE2L2NQO2PTGS1APPHSD11B1
SCHEMBL8462151 0.73 XDH (0.47) APPFBP1
SCHEMBL22468800 0.71 NFE2L2 (0.78) NFE2L2NQO2PTGS1APPHSD11B1
SCHEMBL700051 0.71 NFE2L2 (0.78) NFE2L2NQO2PTGS1APPHSD11B1
SCHEMBL13766470 0.71 NFE2L2 (0.78) NFE2L2NQO2PTGS1APPHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4165023-A1 INHIBITORS OF APOL1 AND USE OF THE SAME Vertex Pharmaceuticals Incorporated (US) 2023-04-19 EP disclosed
CN-115867532-A Inhibitors of APOL1 and uses thereof 弗特克斯药品有限公司 2023-03-28 CN disclosed
EP-0743938-B1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 1999-04-21 EP disclosed