SCHEMBL8387002

SCHEMBL8387002

CCCC=C(CC)C(=O)OOC(=O)C(=CCCC)CC.O=C(Cc1ccccc1I)OOC(=O)Cc1ccccc1I

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPK8 P45983 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8387001 0.93 CYP1A2 (0.35) CYP1A2CYP2D6CYP2C9CYP2C19MAPK8
SCHEMBL3501336 0.78 CYP1A2 (0.53) CYP1A2CYP2D6CYP2C9CYP2C19MAPK8
SCHEMBL7655562 0.74 GRIK1 (0.40)
SCHEMBL7655559 0.74 GRIK1 (0.40)
SCHEMBL2311723 0.69 ALDH1A1 (0.47) CYP1A2CYP2D6CYP2C9CYP2C19PKM
SCHEMBL5132516 0.69 PKM (0.56) CYP1A2CYP2D6CYP2C9CYP2C19PKM
SCHEMBL3623804 0.68 CYP1A2 (0.54) CYP1A2CYP2D6CYP2C9CYP2C19MAPK8
SCHEMBL30776972 0.68 CYP1A2 (0.54) CYP1A2CYP2D6CYP2C9CYP2C19MAPK8
SCHEMBL21635610 0.66 CYP1A2 (0.51) CYP1A2CYP2D6CYP2C9CYP2C19MAPK8
SCHEMBL2315505 0.66 TSHR (0.51) CYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0907666-A1 PARTICLES COMPRISING AMPHIPHILIC COPOLYMERS, HAVING A CROSS-LINKED SHELL DOMAIN AND AN INTERIOR CORE DOMAIN, USEFUL FOR PHARMACEUTICAL AND OTHER APPLICATIONS G.D. Searle & Co. (US) 1999-04-14 EP disclosed
WO-1997049736-A2 PARTICLES COMPRISING AMPHIPHILIC COPOLYMERS, HAVING A CROSS-LINKED SHELL DOMAIN AND AN INTERIOR CORE DOMAIN, USEFUL FOR PHARMACEUTICAL AND OTHER APPLICATIONS G.D. SEARLE AND CO. (US) 1997-12-31 WO disclosed