SCHEMBL8395657

SCHEMBL8395657

CCOCCCN1CCN(CCOC)C1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 4/20 0.41
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM4E B2RXH2 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HSD11B1 P28845 1/20 0.33
HRH2 P25021 1/20 0.31
HTT P42858 1/20 0.30
MAPK1 P28482 1/20 0.30
RAB9A P51151 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GBA1 P04062 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10926779 0.86 HRH1 (0.41) HRH1CYP2D6CYP2C19KDM4ETDP1
SCHEMBL13612608 0.86 HRH1 (0.46) HRH1CYP2D6CYP2C19KDM4EHSD11B1
SCHEMBL10961176 0.84 CYP2D6 (0.41) HRH1CYP2D6CYP2C19KDM4ETDP1
SCHEMBL29322718 0.82 MAPK1 (0.40) CYP2D6CYP2C19KDM4ETDP1MAPK1
SCHEMBL8583237 0.82 ALDH1A1 (0.36) HRH1CYP2D6CYP2C19KDM4ETDP1
SCHEMBL11569854 0.82
SCHEMBL10960846 0.79 HRH3 (0.39) HRH1KDM4EHSD11B1MAPK1RAB9A
SCHEMBL10930283 0.78 HSD11B1 (0.42) KDM4EHSD11B1MAPK1RAB9AALDH1A1
SCHEMBL329951 0.77 LMNA (0.32) HRH1CYP2D6CYP2C19KDM4ETDP1
SCHEMBL11572427 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2901297-B2 1999-06-07 JP claimed
EP-0378657-A1 OXAZOLIDINONE PENETRATION ENHANCING COMPOUNDS. RAJADHYAKSHA VITHAL J 1990-07-25 EP claimed
WO-1990000407-A1 OXAZOLIDINONE PENETRATION ENHANCING COMPOUNDS RAJADHYAKSHA VITHAL J (US) 1990-01-25 WO claimed