SCHEMBL8396192

SCHEMBL8396192

CCCCNc1cccc(N)n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 8/20 0.58
CHRNB2 P17787 2/20 0.45
CHRNB4 P30926 2/20 0.45
CHRNA3 P32297 2/20 0.45
CHRNA4 P43681 2/20 0.45
TLR7 Q9NYK1 3/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KDM4E B2RXH2 2/20 0.41
HRH3 Q9Y5N1 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
XIAP P98170 1/20 0.41
BIRC2 Q13490 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9299788 0.95 TLR8 (0.53) TLR8CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL1099019 0.81 CACNA1C (0.51) ALDH1A1KDM4ENPSR1XIAPBIRC2
SCHEMBL516003 0.81 TLR8 (0.51) TLR8CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL11721783 0.80 TLR8 (0.51) TLR8CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL16790977 0.79 HRH3 (0.43) ALDH1A1TSHRKDM4EHRH3XIAP
SCHEMBL6469127 0.78 TLR8 (0.53) TLR8TLR7ALDH1A1LMNATP53
SCHEMBL22011153 0.78 HRH4 (0.40) TLR8ALDH1A1KDM4EHRH3XIAP
SCHEMBL1099121 0.78 KDM4E (0.46) ALDH1A1LMNAMAPK1KDM4EXIAP
Hydrochloric Acid SCHEMBL16766687 0.78 ALDH1A1 (0.44) ALDH1A1TSHRKDM4EHRH3XIAP
SCHEMBL3222006 0.77 HRH3 (0.59) ALDH1A1HRH3XIAPBIRC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939553-A Process for preparing pyridine-2,6-diamines AKZO NOBEL N.V. (NL) 1999-08-17 US disclosed
EP-0825985-B1 A PROCESS FOR PREPARING PYRIDINE-2,6-DIAMINES AKZO NOBEL NV (NL) 1999-05-26 EP disclosed
EP-0825985-A1 A PROCESS FOR PREPARING PYRIDINE-2,6-DIAMINES Akzo Nobel N.V. (NL) 1998-03-04 EP disclosed
WO-1996036607-A1 A PROCESS FOR PREPARING PYRIDINE-2,6-DIAMINES AKZO NOBEL N.V. (NL) 1996-11-21 WO disclosed