SCHEMBL8397188

SCHEMBL8397188

O=C(NC(=O)[C@@H]1CCCN1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSC P53634 2/20 0.49
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
HTR2C P28335 2/20 0.47
HTR2B P41595 2/20 0.47
HDAC1 Q13547 1/20 0.46
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C19 P33261 1/20 0.45
MC4R P32245 1/20 0.44
GAA P10253 1/20 0.43
ATM Q13315 1/20 0.43
ELANE P08246 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11242758 0.92 CYP1A2 (0.49) NPC1RAB9AHDAC1CYP1A2MC4R
SCHEMBL14490487 0.83 HTT (0.53) HDAC1GAATSHR
SCHEMBL7511740 0.83 GPR6 (0.46) NPC1RAB9AHTR2CHTR2BHDAC1
SCHEMBL1467298 0.82 CTSC (0.53) CTSCNPC1RAB9AHTR2CHTR2B
Hydrochloric Acid SCHEMBL15251815 0.81 CTSC (0.52) CTSCNPC1RAB9AHTR2CHTR2B
SCHEMBL8393442 0.81 DPP4 (0.54) CYP2C19
SCHEMBL8535632 0.81 DPP4 (0.54) CYP2C19
SCHEMBL13570366 0.80 GPR6 (0.49) NPC1RAB9AGAATSHR
Hydrochloric Acid SCHEMBL27541624 0.80 DPP4 (0.54)
SCHEMBL168919 0.78 ELANE (0.54) CTSCNPC1RAB9AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915908-A1 DOLASTATIN PENTAPEPTIDE DERIVATIVES AND THEIR USE AS ANTITUMOR AGENTS BASF AKTIENGESELLSCHAFT (DE) 1999-05-19 EP disclosed
WO-1998004581-A1 DOLASTATIN PENTAPEPTIDE DERIVATIVES AND THEIR USE AS ANTITUMOR AGENTS BASF AKTIENGESELLSCHAFT (DE) 1998-02-05 WO disclosed