SCHEMBL839970

SCHEMBL839970

CCCC(=O)N(CCNC(=O)[C@@H](CS)CC(C)C)Cc1ccc(-c2ccccc2S(=O)(=O)NC(C)=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 10/20 0.42
AGTR2 P50052 2/20 0.42
MME P08473 8/20 0.38
LTB4R2 Q9NPC1 2/20 0.37
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL841556 0.95 LTB4R2 (0.42) AGTR1AGTR2MMELTB4R2
SCHEMBL839509 0.93 AGTR1 (0.43) AGTR1AGTR2MMELTB4R2OPRM1
SCHEMBL841734 0.90 AGTR1 (0.46) AGTR1AGTR2MMELTB4R2
SCHEMBL841733 0.90 AGTR1 (0.46) AGTR1AGTR2MMELTB4R2
SCHEMBL840212 0.89 AGTR1 (0.36) AGTR1AGTR2MME
SCHEMBL840307 0.89 AGTR1 (0.41) AGTR1AGTR2MMELTB4R2
SCHEMBL840866 0.88 AGTR1 (0.43) AGTR1AGTR2MMELTB4R2
SCHEMBL839461 0.87 AGTR1 (0.43) AGTR1AGTR2LTB4R2
SCHEMBL839460 0.87 AGTR1 (0.43) AGTR1AGTR2LTB4R2
SCHEMBL859395 0.86 LTB4R2 (0.47) AGTR1AGTR2MMELTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143298-B2 Dual-acting antihypertensive agents THERAVANCE, INC. (US) 2012-03-27 US disclosed