SCHEMBL8399991

SCHEMBL8399991

COc1ccc(-c2c(NCCN3CCCCC3)cc3cc(OC)ccc3c2Oc2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 8/20 0.54
ESR1 P03372 4/20 0.50
ESR2 Q92731 1/20 0.43
SMARCA2 P51531 1/20 0.43
BACE1 P56817 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8399940 0.99 ACP1 (0.53) ACP1ESR1ESR2SMARCA2BACE1
SCHEMBL8399903 0.95 ACP1 (0.49) ACP1ESR1ESR2
SCHEMBL8403143 0.93 ACP1 (0.55) ACP1ESR1ESR2SMARCA2
SCHEMBL8401756 0.93 ESR1 (0.51) ACP1ESR1ESR2
SCHEMBL8405723 0.87 ACP1 (0.49) ACP1ESR1ESR2SMARCA2
SCHEMBL8403332 0.86 ESR1 (0.54) ACP1ESR1ESR2SMARCA2
SCHEMBL8519431 0.85 ESR1 (0.52) ESR1ESR2
SCHEMBL8400248 0.83 KMT2A (0.53) ESR1
SCHEMBL8403608 0.83 ESR1 (0.50) ACP1ESR1ESR2SMARCA2
SCHEMBL8400253 0.83 ESR1 (0.47) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929090-A NOVEL COMPOUNDS FOR TREATING ESTROGEN DEPRIVATION CAUSED BY MENOPAUSE OR OVARIECTOMY; TREATING OSTEOPOROSIS, CARDIOVASCULAR DISEASES, AND ENDOMETRIOSIS ELI LILLY AND COMPANY (US) 1999-07-27 US disclosed