SCHEMBL8400136

SCHEMBL8400136

CN(C)CCON.ClOCl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRM2 P08172 2/20 0.36
CHRM4 P08173 2/20 0.36
CHRM5 P08912 2/20 0.36
CHRM1 P11229 2/20 0.36
CHRM3 P20309 2/20 0.36
MAPT P10636 2/20 0.35
CA12 O43570 3/20 0.34
CA2 P00918 3/20 0.34
CA9 Q16790 3/20 0.34
CA1 P00915 2/20 0.34
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
TSHR P16473 2/20 0.32
ALDH1A1 P00352 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2126204 0.91
Hydrochloric Acid SCHEMBL2789718 0.88
Hydrochloric Acid SCHEMBL3892675 0.88
Cyclopropane SCHEMBL28089739 0.83 CHRM2 (0.36) CHRNB2CHRNA4CHRM2CHRM4CHRM5
SCHEMBL6207154 0.74
Hydrochloric Acid SCHEMBL8413000 0.72 ADRB2 (0.46) ADRB2ADRB1ADRB3TSHRALDH1A1
Hydrochloric Acid SCHEMBL5074625 0.72 ADRB2 (0.46) ADRB2ADRB1ADRB3TSHRALDH1A1
Hydrochloric Acid SCHEMBL4960594 0.72
SCHEMBL28522463 0.72 CA12 (0.50) CHRNB2CHRNA4CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL8415270 0.70 ALDH1A1 (0.50) ADRB2ADRB1ADRB3TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0742214-B1 Seco-D steroids active in the cardiovascular system and pharmaceutical compositions containing same SIGMA TAU IND FARMACEUTI (IT) 1999-06-16 EP disclosed
US-5731345-A Seco-D steroids active on the cardiovascular system and pharmaceutical compositions containing same SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A (IT) 1998-03-24 US disclosed