SCHEMBL8401715

SCHEMBL8401715

CCCNC(=C[N+](=O)[O-])N(C)Cc1ccc(Cl)nc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.38
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 4/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
CHRNA1 P02708 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA7 P36544 1/20 0.35
HSP90AA1 P07900 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CASP6 P55212 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3282952 0.91 ALDH1A1 (0.38) FAAHCHRNB2CHRNA4SMN1; SMN2ALDH1A1
SCHEMBL7106155 0.86 CHRNB2 (0.39) CHRNB2CHRNA4SMN1; SMN2ALDH1A1CYP3A4
SCHEMBL5001742 0.86 CHRNB2 (0.39) CHRNB2CHRNA4SMN1; SMN2ALDH1A1CYP3A4
SCHEMBL8405273 0.85 ALDH1A1 (0.36) FAAHCHRNB2CHRNA4SMN1; SMN2ALDH1A1
SCHEMBL8404142 0.84 CHRNB2 (0.38) CHRNB2CHRNA4SMN1; SMN2ALDH1A1CYP3A4
SCHEMBL8405604 0.83 CHRNA1 (0.38) CHRNB2CHRNA4SMN1; SMN2ALDH1A1CYP3A4
SCHEMBL2801383 0.82 FAAH (0.43) FAAHCHRNB2CHRNA4SMN1; SMN2ALDH1A1
SCHEMBL7662120 0.82 ALDH1A1 (0.36) FAAHCHRNB2CHRNA4SMN1; SMN2ALDH1A1
SCHEMBL888609 0.82 FAAH (0.43) FAAHCHRNB2CHRNA4SMN1; SMN2ALDH1A1
SCHEMBL1747891 0.81 FAAH (0.40) FAAHCHRNB2CHRNA4SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935981-A INSECTICIDAL/MITICIDAL ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-08-10 US disclosed
US-5849768-A α-unsaturated amines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-12-15 US disclosed