SCHEMBL8403348

SCHEMBL8403348

Oc1ccc2nc(O)nnc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
ENPP2 Q13822 1/20 0.45
SRC P12931 1/20 0.43
MEN1 O00255 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
KMT2A Q03164 1/20 0.41
ESR2 Q92731 8/20 0.38
ESR1 P03372 6/20 0.38
HTT P42858 2/20 0.38
PLAU P00749 1/20 0.38
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TTR P02766 1/20 0.35
PIK3CG P48736 1/20 0.35
PABPC1 P11940 1/20 0.35
ESRRB O95718 1/20 0.35
ESRRA P11474 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15293604 0.78 ALDH1A1 (0.42) ALDH1A1KDM4EHPGDENPP2SRC
SCHEMBL8404114 0.78 PIK3CG (0.60) ALDH1A1KDM4EMEN1KMT2APIK3CG
SCHEMBL8749320 0.78 NQO2 (0.52) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL3532558 0.78 SRC (0.67) ALDH1A1KDM4EHPGDENPP2SRC
SCHEMBL14077239 0.78 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDENPP2MEN1
SCHEMBL2368334 0.78 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDENPP2MEN1
SCHEMBL8399923 0.74 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL8749540 0.74 TRPA1 (0.44) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL14582918 0.73 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDENPP2MEN1
SCHEMBL6243628 0.73 PDPK1 (0.52) ALDH1A1KDM4EHPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856325-A REDUCING INFLAMMATION BY INHIBITING PLA2 IN A MAMMAL BOEHRINGER MANNHEIM GMBH (DE) 1999-01-05 US disclosed
EP-0675881-B1 Use of benzotriazines as PLA2-Inhibitors and new benzotriazines BOEHRINGER MANNHEIM GMBH (DE) 1997-03-19 EP disclosed