SCHEMBL840514

SCHEMBL840514

[CH2]c1ccc(NC=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.45
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL469386 0.86 ALDH1A1 (0.72) ALDH1A1LMNAMEN1KMT2A
SCHEMBL28553974 0.79 ALDH1A1 (0.56) ALDH1A1LMNAMEN1KMT2A
SCHEMBL838486 0.78 ALDH1A1 (0.50) ALDH1A1LMNAMEN1KMT2A
SCHEMBL9472659 0.76 ALDH1A1 (0.59) ALDH1A1LMNAMEN1KMT2A
SCHEMBL1451254 0.75 ALDH1A1 (0.52) ALDH1A1LMNAMEN1KMT2A
SCHEMBL90440 0.74 ALDH1A1 (0.56) ALDH1A1LMNAMEN1KMT2A
SCHEMBL515529 0.74 ALDH1A1 (0.56) ALDH1A1LMNAMEN1KMT2A
SCHEMBL14605366 0.74 ALDH1A1 (0.56) ALDH1A1LMNAMEN1KMT2A
SCHEMBL428217 0.74 ALDH1A1 (0.56) ALDH1A1LMNAMEN1KMT2A
SCHEMBL4457780 0.74 ALDH1A1 (0.56) ALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0145304-B1 TETRAHYDRO-BETA-CARBOLINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Tanabe Seiyaku Co., Ltd. (JP) 1988-04-20 EP claimed
EP-0128021-B1 TETRAHYDRO-BETA-CARBOLINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Tanabe Seiyaku Co., Ltd. (JP) 1987-09-09 EP claimed
US-4628057-A Tetrahydro-β-carboline derivatives and treatment of liver diseases TANABE SEIYAKU CO., LTD. (JP) 1986-12-09 US claimed
US-4612317-A Tetrahydro-β-carboline dithioic acid derivatives and treatment of liver diseases TANABE SEIYAKU CO., LTD. (JP) 1986-09-16 US claimed
EP-0145304-A1 Tetrahydro-beta-carboline derivatives and process for the preparation thereof Tanabe Seiyaku Co., Ltd. (JP) 1985-06-19 EP claimed
EP-0128021-A1 Tetrahydro-beta-carboline derivatives and process for the preparation thereof Tanabe Seiyaku Co., Ltd. (JP) 1984-12-12 EP claimed
EP-1493819-B1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER UBE INDUSTRIES (JP) 2014-11-12 EP disclosed
US-8143052-B2 Process for preparing optically active (S or R)-α amino acid and (R or S)-α amino acid ester in one phase organic reaction medium UBE INDUSTRIES, LTD. (JP) 2012-03-27 US disclosed
US-7915019-B2 Processes for preparing optically active (S or R)-β-amino acid and optically active (R or S)-β-amino acid ester, and β-amino acid 2-alkoxyethyl ester and optically active (S or R)-β amino acid 2-alkoxyethyl ester UBE INDUSTRIES, LTD. (JP) 2011-03-29 US disclosed
EP-1840218-B1 Process for production of optically active (S)- or (R)-beta-amino acids and optically active (R)- or (S)-beta -amino acid esters, and optically active (S)- or (R)-2-alkoxyethyl esters of beta-amino acids. UBE INDUSTRIES (JP) 2011-02-23 EP disclosed
US-20090117626-A1 Process for preparing carboxylic acid using surfactant-modified enzyme UBE INDUSTRIES, LTD. (JP) 2009-05-07 US disclosed
US-20090042260-A1 PROCESS FOR PREPARING OPTICALLY ACTIVE (S OR R)-ALPHA-AMINO ACID AND OPTICALLY ACTIVE (R OR S)-ALPHA-AMINO ACID ESTER UBE INDUSTRIES, LTD. (JP) 2009-02-12 US disclosed
US-7449325-B2 Process for enzymatically producing either optically active N-substituted β-amino acids or esters thereof or optically active N-substituted 2-homopipecolic acids or esters thereof UBE INDUSTRIES, LTD. (JP) 2008-11-11 US disclosed
EP-0676398-A2 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1995-10-11 EP disclosed
EP-0145304-B1 TETRAHYDRO-BETA-CARBOLINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Tanabe Seiyaku Co., Ltd. (JP) 1988-04-20 EP disclosed
EP-0128021-B1 TETRAHYDRO-BETA-CARBOLINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Tanabe Seiyaku Co., Ltd. (JP) 1987-09-09 EP disclosed
US-4628057-A Tetrahydro-β-carboline derivatives and treatment of liver diseases TANABE SEIYAKU CO., LTD. (JP) 1986-12-09 US disclosed
US-4612317-A Tetrahydro-β-carboline dithioic acid derivatives and treatment of liver diseases TANABE SEIYAKU CO., LTD. (JP) 1986-09-16 US disclosed
EP-0145304-A1 Tetrahydro-beta-carboline derivatives and process for the preparation thereof Tanabe Seiyaku Co., Ltd. (JP) 1985-06-19 EP disclosed
EP-0128021-A1 Tetrahydro-beta-carboline derivatives and process for the preparation thereof Tanabe Seiyaku Co., Ltd. (JP) 1984-12-12 EP disclosed