SCHEMBL8406480

SCHEMBL8406480

CC(C)N(c1ncccc1[N+](=O)[O-])C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.53
DRD4 P21917 3/20 0.53
DRD3 P35462 3/20 0.53
ALDH1A1 P00352 3/20 0.53
GMNN O75496 2/20 0.53
LMNA P02545 2/20 0.53
HPGD P15428 2/20 0.53
PMP22 Q01453 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
TDP1 Q9NUW8 2/20 0.53
TP53 P04637 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
MAPK1 P28482 3/20 0.49
SIGMAR1 Q99720 2/20 0.48
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.45
OPRM1 P35372 1/20 0.44
DRD1 P21728 1/20 0.44
HTR2A P28223 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8409521 0.86 DRD2 (0.61) DRD2DRD4DRD3ALDH1A1GMNN
SCHEMBL8409570 0.84 MAPK1 (0.50) DRD2DRD4DRD3ALDH1A1GMNN
SCHEMBL8408645 0.83 MAPK1 (0.51) DRD2DRD4DRD3ALDH1A1GMNN
SCHEMBL8791696 0.83 MAPK1 (0.48) DRD2DRD4DRD3ALDH1A1GMNN
SCHEMBL8408436 0.82 DRD2 (0.58) DRD2DRD4DRD3ALDH1A1GMNN
SCHEMBL8406813 0.81 LMNA (0.48) DRD2DRD4DRD3ALDH1A1GMNN
SCHEMBL8792951 0.79 DRD2 (0.58) DRD2DRD4DRD3ALDH1A1GMNN
SCHEMBL8406474 0.79 DRD2 (0.55) DRD2DRD4DRD3ALDH1A1GMNN
SCHEMBL8406930 0.79 MAPK1 (0.48) MAPK1SIGMAR1KMT2APOLBMEN1
SCHEMBL8406471 0.78 DRD2 (0.54) DRD2DRD4DRD3ALDH1A1GMNN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866589-A Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds PHARMACIA & UPJOHN COMPANY (US) 1999-02-02 US disclosed
EP-0797576-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1997-10-01 EP disclosed
WO-1996018628-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-06-20 WO disclosed