SCHEMBL8406780

SCHEMBL8406780

O=Cc1ccc(O)c(CCc2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.48
PTGS2 P35354 2/20 0.48
RAB9A P51151 1/20 0.48
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
ALOX15 P16050 4/20 0.44
CYP3A4 P08684 3/20 0.44
HSD17B10 Q99714 3/20 0.44
HPGD P15428 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
HIF1A Q16665 2/20 0.44
BCL2 P10415 1/20 0.43
BCL2L1 Q07817 1/20 0.43
ALDH1A1 P00352 3/20 0.43
ALOX12 P18054 2/20 0.43
MAPK1 P28482 2/20 0.43
EGFR P00533 2/20 0.43
LCK P06239 2/20 0.43
TDP1 Q9NUW8 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9487127 0.78 ALOX15 (0.60) KDM4EPTGS2ALOX15CYP3A4HSD17B10
SCHEMBL14540315 0.78 KDM4E (0.46) KDM4EPTGS2RAB9AALOX15CYP3A4
SCHEMBL3429484 0.77 KDM4E (0.53) KDM4EPTGS2RAB9AHPGDALDH1A1
SCHEMBL1426624 0.77 EGFR (0.60) ALOX15CYP3A4HSD17B10HPGDHIF1A
SCHEMBL9243499 0.77 BACE1 (0.50) KDM4EALOX15CYP3A4HSD17B10HPGD
SCHEMBL18519791 0.77 ALDH1A1 (0.48) MAOAMAOBHPGDMEN1KMT2A
SCHEMBL13144543 0.76 NPSR1 (0.59) RAB9AHPGDMEN1KMT2AALDH1A1
SCHEMBL7507833 0.76 KDM4E (0.61) KDM4EPTGS2RAB9AALOX15CYP3A4
SCHEMBL17982835 0.76 CA1 (0.61) KDM4EALOX15HPGDMEN1KMT2A
SCHEMBL9156902 0.76 BCL2 (0.58) KDM4EMAOAMAOBALOX15BCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0778821-B1 ORTHO-SUBSTITUTED AROMATIC ETHER COMPOUNDS AND THEIR USE IN PHARMACEUTICAL COMPOSITIONS FOR PAIN RELIEF ZENECA LTD (GB) 1999-10-20 EP disclosed
US-5965741-A ANTIINFLAMMATORY, ANTIPYRETIC AND ANTIDIARRHOEAL PROPERTIES ZENECA LIMITED (GB) 1999-10-12 US disclosed
EP-0778821-A1 ORTHO-SUBSTITUTED AROMATIC ETHER COMPOUNDS AND THEIR USE IN PHARMACEUTICAL COMPOSITIONS FOR PAIN RELIEF ZENECA LIMITED (GB) 1997-06-18 EP disclosed
WO-1996006822-A1 ORTHO-SUBSTITUTED AROMATIC ETHER COMPOUNDS AND THEIR USE IN PHARMACEUTICAL COMPOSITIONS FOR PAIN RELIEF ZENECA LIMITED (GB) 1996-03-07 WO disclosed