SCHEMBL8407196

SCHEMBL8407196

Fc1ccc(Oc2ccc(F)c(CBr)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FDFT1 P37268 3/20 0.46
FFAR4 Q5NUL3 2/20 0.39
SOS1 Q07889 3/20 0.38
HSPB1 P04792 1/20 0.38
HTR2A P28223 4/20 0.36
SLC6A4 P31645 4/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
KCNH2 Q12809 3/20 0.36
CACNA1C Q13936 1/20 0.36
LTA4H P09960 2/20 0.36
SCN4A P35499 1/20 0.34
EPHX2 P34913 1/20 0.34
FFAR1 O14842 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11383668 0.87 LTA4H (0.43) FFAR4HTR2ASLC6A4LTA4HFFAR1
SCHEMBL11292143 0.84 FFAR4 (0.43) FFAR4SLC6A4KCNH2FFAR1
SCHEMBL2294122 0.84 SOS1 (0.41) FDFT1FFAR4SOS1HSPB1HTR2A
SCHEMBL11326273 0.81 FDFT1 (0.46) FDFT1FFAR4SOS1HSPB1PDE4A
SCHEMBL4371661 0.79 HTR2A (0.44) SOS1HTR2ASLC6A4KCNH2
SCHEMBL119218 0.78 DPP4 (0.46)
SCHEMBL29430341 0.78 DPP4 (0.46)
SCHEMBL378823 0.77 MTNR1B (0.51) HTR2A
SCHEMBL31051591 0.77 MTNR1B (0.51) HTR2A
SCHEMBL11029838 0.76 DPP4 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5872137-A AROMATIC OXY DIHALOPRENE COMPOUNDS INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-02-16 US disclosed
EP-0722430-B1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL CO (JP) 1998-10-21 EP disclosed
EP-0722430-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-07-24 EP disclosed
WO-1996004228-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-02-15 WO disclosed