SCHEMBL119218

SCHEMBL119218

Fc1ccc(F)c(CBr)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.46
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
CA3 P07451 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
IDO1 P14902 2/20 0.39
AGXT P21549 2/20 0.39
RIPK1 Q13546 2/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
DPP8 Q6V1X1 2/20 0.38
MAPK8 P45983 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29430341 1.00 DPP4 (0.46) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL11029838 0.98 DPP4 (0.44) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL5038406 0.98 DPP4 (0.44) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL3307736 0.82 IDO1 (0.40) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL30149750 0.82 IDO1 (0.40) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL27830893 0.81 DPP4 (0.43) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL29453657 0.80 IDO1 (0.54) CA3CA6CA5ACA9CA14
SCHEMBL120150 0.80 IDO1 (0.54) CA3CA6CA5ACA9CA14
SCHEMBL5252643 0.79 MPO (0.49) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL7700255 0.79 CA3 (0.46) DPP4PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 831 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116640106-B Phenylpiperazine compound and preparation method and application thereof 郑州大学 2024-03-08 CN claimed
CN-117586257-A Compound containing 2, 8-diazaspiro [4.5] decan-1-one skeleton and application thereof 中国药科大学 2024-02-23 CN claimed
CN-116640106-A Phenylpiperazine compound and preparation method and application thereof 郑州大学 2023-08-25 CN claimed
US-20080177077-A1 PROCESSES FOR THE PREPARATION OF 3-(4-(2,4-DIFLUOROBENZYLOXY)-3-BROMO-6-METHYL-2-OXOPYRIDIN-1(2H)-YL)-N,4-DIMETHYLBENZAMIDE PFIZER, INC. 2008-07-24 US claimed
US-12617880-B2 Compounds for use in catalyst compositions for the production of polyolefins SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2026-05-05 US disclosed
EP-3966226-B1 MASP INHIBITORY COMPOUNDS AND USES THEREOF BAYER AG (DE) 2025-12-24 EP disclosed
US-12503491-B2 MASP inhibitory compounds and uses thereof BAYER AKTIENGESELLSCHAFT (DE) 2025-12-23 US disclosed
EP-4605394-A1 PYRIMIDINE SGC STIMULATORS Tisento Therapeutics Inc. (US) 2025-08-27 EP disclosed
US-20250243205-A1 sGC STIMULATORS TISENTO THERAPEUTICS INC (US) 2025-07-31 US disclosed
US-12331056-B2 SHP2 phosphatase inhibitors and methods of use thereof RELAY THERAPEUTICS, INC. (US) 2025-06-17 US disclosed
US-12281101-B2 Bicyclic lactams and methods of use thereof GENENTECH, INC. (US) 2025-04-22 US disclosed
US-20250122171-A1 Substituted Amine Compounds, Compositions and Methods of Use DEEP APPLE THERAPEUTICS, INC. 2025-04-17 US disclosed
US-5352678-A Dopaminergic agents BRISTOL-MYERS SQUIBB CO. (US) 1994-10-04 US disclosed
EP-0594573-A1 PREPARATION OF PROPENOIC ACID DERIVATIVES AgrEvo UK Limited (GB) 1994-05-04 EP disclosed
US-5264609-A Etherification and hydrolysis SCHERING AGROCHEMICALS LIMITED (GB) 1993-11-23 US disclosed
EP-0546583-A1 Piperazinyl-and piperidinyl-cyclohexanols Bristol-Myers Squibb Company (US) 1993-06-16 EP disclosed
WO-1991007385-A1 PREPARATION OF PROPENOIC ACID DERIVATIVES SCHERING AGROCHEMICALS LIMITED (GB) 1991-05-30 WO disclosed
US-4695579-A Antifungal 2-azolylmethyl-3-difluorobenzyloxy-2,3-dihydrofluoro-benzo(B) thiophens SCHERING CORPORATION (US) 1987-09-22 US disclosed
EP-0185381-A2 2-Azolylmethyl-3-difluorobenzyloxy-2,3-dihydrofluorobenzo(b)thiophenes, process for their preparation and compositions containing them SCHERING CORPORATION (US) 1986-06-25 EP disclosed
EP-0157637-A2 Heterocyclic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1985-10-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12503491-B2 MASP inhibitory compounds and uses thereof MASP2, SERPINB1, SPINT2 DPP4 109/4885PSEN1 4382/4885PSEN2 4657/4885
US-12617880-B2 Compounds for use in catalyst compositions for the production of polyolefins PRMT5, CBR3, MET DPP4 4636/4885PSEN1 4753/4885PSEN2 4736/4885
US-20250122171-A1 Substituted Amine Compounds, Compositions and Methods of Use MRGPRX2, MRGPRX1, MRGPRX4 DPP4 2501/4885PSEN1 2497/4885PSEN2 1073/4885
US-12281101-B2 Bicyclic lactams and methods of use thereof LSS, LPXN, CYP1B1 DPP4 3964/4885PSEN1 263/4885PSEN2 1218/4885
US-20250243205-A1 sGC STIMULATORS GMPS, GUCY1A2, PDE2A DPP4 2780/4885PSEN1 3549/4885PSEN2 3765/4885
US-20080177077-A1 PROCESSES FOR THE PREPARATION OF 3-(4-(2,4-DIFLUOROBENZYLOXY)-3-BROMO-6-METHYL-2-OXOPYRIDIN-1(2H)-YL)-N,4-DIMETHYLBENZAMIDE CYP4X1, CYP4B1, KDM4B DPP4 871/4885PSEN1 3711/4885PSEN2 2463/4885
US-12331056-B2 SHP2 phosphatase inhibitors and methods of use thereof PTPRCAP, PTPN22, PTPN1 DPP4 2451/4885PSEN1 3200/4885PSEN2 2745/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.