SCHEMBL8409274

SCHEMBL8409274

O=C(Cl)c1cccc(Cl)c1O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
KLKB1 P03952 1/20 0.49
TSHR P16473 3/20 0.48
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
PLAU P00749 2/20 0.45
PLAT P00750 2/20 0.45
F2 P00734 1/20 0.45
F10 P00742 1/20 0.45
P2RX1 P51575 1/20 0.45
P2RX4 Q99571 1/20 0.45
P2RX7 Q99572 1/20 0.45
TMPRSS4 Q9NRS4 1/20 0.45
ALOX15 P16050 2/20 0.45
POLB P06746 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL236867 0.85 ALDH1A1 (0.52) ALDH1A1TSHRCES2CES1ALOX15
SCHEMBL29499766 0.82 TSHR (0.65) ALDH1A1KLKB1TSHRCES2CES1
SCHEMBL372307 0.82 TSHR (0.65) ALDH1A1KLKB1TSHRCES2CES1
SCHEMBL3607272 0.81 KLKB1 (0.61) ALDH1A1KLKB1PLAUPLATF2
SCHEMBL431965 0.80 TSHR (0.63) ALDH1A1KLKB1TSHRCES2CES1
SCHEMBL10779351 0.80 TSHR (0.63) ALDH1A1KLKB1TSHRCES2CES1
SCHEMBL425111 0.80 TSHR (0.63) ALDH1A1KLKB1TSHRCES2CES1
SCHEMBL30779693 0.80 KLKB1 (0.51) ALDH1A1KLKB1TSHRCES2CES1
SCHEMBL421701 0.80 KLKB1 (0.51) ALDH1A1KLKB1TSHRCES2CES1
SCHEMBL2522829 0.80 KLKB1 (0.51) ALDH1A1KLKB1TSHRCES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108395406-A A kind of benzimidazolone AS-BI production technologies 中卫市创科知识产权投资有限公司 2018-08-14 CN claimed
CN-108395406-A A kind of benzimidazolone AS-BI production technologies 中卫市创科知识产权投资有限公司 2018-08-14 CN disclosed
CN-103275034-B Preparation method of micromolecule cathepsin D inhibitor NANJING UNIVERSITY OF TECHNOLOGY 2015-07-08 CN disclosed
CN-103992336-A Oxa- or thio-evodiamine anti-tumor derivatives and preparation method thereof UNIV PLA 2ND MILITARY MEDICAL 2014-08-20 CN disclosed
CN-103275034-A Preparation method of micromolecule cathepsin D inhibitor NANJING UNIVERSITY OF TECHNOLOGY 2013-09-04 CN disclosed
CN-102206152-A Method for chemically synthesizing 3,5-diio-2-hydroxybenzene formyl chloride ZHEJIANG RONGYAO CHEMICAL CO LTD 2011-10-05 CN disclosed
EP-0778821-B1 ORTHO-SUBSTITUTED AROMATIC ETHER COMPOUNDS AND THEIR USE IN PHARMACEUTICAL COMPOSITIONS FOR PAIN RELIEF ZENECA LTD (GB) 1999-10-20 EP disclosed
US-5965741-A ANTIINFLAMMATORY, ANTIPYRETIC AND ANTIDIARRHOEAL PROPERTIES ZENECA LIMITED (GB) 1999-10-12 US disclosed
EP-0778821-A1 ORTHO-SUBSTITUTED AROMATIC ETHER COMPOUNDS AND THEIR USE IN PHARMACEUTICAL COMPOSITIONS FOR PAIN RELIEF ZENECA LIMITED (GB) 1997-06-18 EP disclosed
WO-1996006822-A1 ORTHO-SUBSTITUTED AROMATIC ETHER COMPOUNDS AND THEIR USE IN PHARMACEUTICAL COMPOSITIONS FOR PAIN RELIEF ZENECA LIMITED (GB) 1996-03-07 WO disclosed