SCHEMBL8409294

SCHEMBL8409294

CCOC(=O)CCCCOc1cc(C)c(N)c(CC)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.45
PDK2 Q15119 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
CYSLTR2 Q9NS75 2/20 0.41
CYSLTR1 Q9Y271 2/20 0.41
LTA4H P09960 3/20 0.40
FFAR1 O14842 1/20 0.40
ALDH2 P05091 2/20 0.40
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
PLA2G2A P14555 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6497458 0.83 BRD4 (0.50) BRD4PDK2CYP1A2CYSLTR2CYSLTR1
SCHEMBL10203017 0.80 BRD4 (0.55) BRD4PDK2CYP4F2CYP4A11CYSLTR2
SCHEMBL6492212 0.77 MAPT (0.46) BRD4PDK2CYP1A2CYSLTR2CYSLTR1
SCHEMBL12975430 0.76 BRD4 (0.57) BRD4PDK2CYSLTR2CYSLTR1LTA4H
SCHEMBL16245544 0.76 LTA4H (0.53) BRD4PDK2CYP1A2CYSLTR2CYSLTR1
SCHEMBL8409159 0.75 LTA4H (0.39) BRD4PDK2CYSLTR2CYSLTR1LTA4H
SCHEMBL3433095 0.74 BRD4 (0.46) BRD4PDK2CYP1A2CYSLTR2CYSLTR1
SCHEMBL17265678 0.74 LTA4H (0.52) BRD4PDK2CYSLTR2CYSLTR1LTA4H
SCHEMBL5457249 0.74 LTA4H (0.52) BRD4PDK2CYSLTR2CYSLTR1LTA4H
SCHEMBL4389091 0.73 BRD4 (0.53) BRD4PDK2CYP1A2CYSLTR2CYSLTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446173-B1 Immunoassay for metolachlorine NOVARTIS AG (CH) 1999-07-14 EP disclosed
US-5576188-A HYBRIDOMA CELL LINE WHICH PRODUCES A MONOCLONAL ANTIBODY HAVING SPECIFIED CHARACTERISTICS CIBA-GEIGY CORPORATION (US) 1996-11-19 US disclosed
EP-0446173-A2 Immunoassay for metolachlorine CIBA-GEIGY AG (CH) 1991-09-11 EP disclosed