SCHEMBL8409477

SCHEMBL8409477

CCCNc1cccnc1N(CC)N1CCNCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.38
KHK P50053 2/20 0.37
HRH4 Q9H3N8 1/20 0.36
FLT3 P36888 1/20 0.35
TYRO3 Q06418 1/20 0.35
MERTK Q12866 1/20 0.35
GAS6 Q14393 1/20 0.35
ALDH1A1 P00352 2/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
ADRA1B P35368 2/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PLD1 Q13393 1/20 0.32
HTR2C P28335 2/20 0.32
HTR3E A5X5Y0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8408425 0.76 SLC6A2 (0.39) PDE5AKHKFLT3TYRO3MERTK
SCHEMBL8917883 0.76 EPHX2 (0.49) KHKHRH4FLT3TYRO3MERTK
SCHEMBL8406794 0.65 SLC6A2 (0.40) ADRA1DADRA1AADRA1BHTR1ASLC6A4
SCHEMBL28884912 0.65 SIGMAR1 (0.42) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL8510998 0.64 PDE5A (0.48) PDE5AALDH1A1ADRA1DADRA1AADRA1B
SCHEMBL1977303 0.64 KDM4E (0.57) PDE5AALDH1A1KDM4EHPGDHSD17B10
SCHEMBL3334093 0.64 EPHX2 (0.51) FLT3TYRO3MERTKGAS6PLD1
SCHEMBL9094827 0.63 SCD (0.38) ALDH1A1TSHRL3MBTL1KDM4EHPGD
SCHEMBL8409833 0.63 KHK (0.37) KHKFLT3TYRO3MERTKGAS6
Hydrochloric Acid SCHEMBL8703350 0.63 EPHX2 (0.50) FLT3TYRO3MERTKGAS6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866589-A Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds PHARMACIA & UPJOHN COMPANY (US) 1999-02-02 US disclosed
WO-1996018628-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-06-20 WO disclosed