SCHEMBL8409849

SCHEMBL8409849

COc1ccc2ccc(OC)c3c2c1CC(NC(C)=O)C3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 6/20 0.66
MTNR1B P49286 5/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8410015 0.89 MTNR1A (0.62) MTNR1AMTNR1B
SCHEMBL8409987 0.80 MTNR1A (1.00) MTNR1AMTNR1B
SCHEMBL11496541 0.80 MTNR1A (0.72) MTNR1AMTNR1B
SCHEMBL8409761 0.79 KDM4E (0.48) MTNR1AMTNR1B
SCHEMBL6081151 0.79 CA1 (0.43) MTNR1AMTNR1B
SCHEMBL6081951 0.78 MTNR1A (0.48) MTNR1AMTNR1B
SCHEMBL6081859 0.78 MTNR1A (0.42) MTNR1AMTNR1B
SCHEMBL7658012 0.76 MTNR1A (0.54) MTNR1AMTNR1B
SCHEMBL8410013 0.76 KDM4E (0.60) MTNR1AMTNR1B
SCHEMBL8407113 0.76 KDM4E (0.46) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737670-B1 Tricyclic amides, processes for their preparation, and pharmaceutical compositions containing them ADIR (FR) 1999-07-21 EP claimed
EP-0737670-B1 Tricyclic amides, processes for their preparation, and pharmaceutical compositions containing them ADIR (FR) 1999-07-21 EP disclosed
US-5849781-A Tricyclic amides ADIR ET COMPAGNIE (FR) 1998-12-15 US disclosed
US-5712312-A MELATONINERGIC RECEPTOR LIGANDS, TREATMENT OF SLEEP DISORDERS ADIR ET COMPAGNIE (FR) 1998-01-27 US disclosed
EP-0737670-A1 Tricyclic amides, processes for their preparation, and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-10-16 EP disclosed