SCHEMBL8410022

SCHEMBL8410022

CC1Cc2cc3c(cc2CN1)OCO3

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 8/20 0.50
ADRA2A P08913 3/20 0.50
ADRA2B P18089 2/20 0.50
ADRA2C P18825 2/20 0.50
ACHE P22303 1/20 0.45
CYP3A4 P08684 2/20 0.42
HTR1A P08908 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX15 P16050 1/20 0.42
NFKB1 P19838 1/20 0.42
MAPK1 P28482 1/20 0.42
CYP2C19 P33261 1/20 0.42
HIF1A Q16665 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11746507 0.82 KDM4E (0.42) ACHECYP3A4HTR1ACYP1A2CYP2D6
SCHEMBL13072958 0.82 PNMT (0.62) PNMTADRA2AADRA2BADRA2C
SCHEMBL11727741 0.74 PNMT (0.54) PNMTADRA2AADRA2BADRA2C
SCHEMBL11727749 0.74 PNMT (0.54) PNMTADRA2AADRA2BADRA2C
SCHEMBL11743824 0.73 ACHE (0.47) ACHECYP3A4HTR1ACYP1A2CYP2D6
SCHEMBL11164603 0.73 EGLN1 (0.44) ACHECYP3A4HTR1AALOX15MAPK1
SCHEMBL1011095 0.72 PNMT (0.51) PNMTADRA2AADRA2BADRA2CACHE
SCHEMBL8410159 0.71 DRD2 (0.44) PNMTADRA2AADRA2BADRA2CCYP3A4
Hydrochloric Acid SCHEMBL11166549 0.71 EGLN1 (0.43) ACHECYP3A4HTR1AALOX15MAPK1
SCHEMBL4689086 0.71 KDM4E (0.42) ACHECYP3A4HTR1ACYP2D6MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919794-A Methods of using pharmaceutical tetrahydroisoquinolines VIRGINIA COMMONWEALTH UNIVERSITY (US) 1999-07-06 US disclosed