SCHEMBL8410099

SCHEMBL8410099

CCNC(=O)c1ccc2c(c1)CN(C(=O)C(Cc1ccc3ccccc3c1)NC(=O)C1CCCCN1C(=O)OC(C)(C)C)C2

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.43
MC5R P33032 1/20 0.43
TACR1 P25103 18/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8412367 0.89 TACR1 (0.45) MC4RMC5RTACR1MAPT
SCHEMBL6163821 0.88 MAPK1 (0.48)
SCHEMBL8410142 0.87 TACR1 (0.52) MC4RMC5RTACR1MAPT
SCHEMBL8412756 0.85 TACR1 (0.51) TACR1
Hydrochloric Acid SCHEMBL6162871 0.80 MC4R (0.46) MC4R
Hydrochloric Acid SCHEMBL6162865 0.80 MC4R (0.46) MC4R
SCHEMBL6161717 0.80 MAPK1 (0.50)
SCHEMBL6161724 0.80 MAPK1 (0.50)
SCHEMBL8412875 0.80 HDAC3 (0.47) TACR1
SCHEMBL6162910 0.79 MAPK1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5936089-A PIPERIDINE DERIVATIVES; BONE DISORDERS; OBESITY; AGING; CACHEXIA ASSOCIATED WITH AIDS AND CANCER PFIZER INC (US) 1999-08-10 US disclosed