SCHEMBL8413899

SCHEMBL8413899

CCCCOc1ccc(OCCCNC(C)C)c(C=O)c1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.53
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
KDM4E B2RXH2 4/20 0.44
RAB9A P51151 1/20 0.44
HTR1B P28222 1/20 0.43
NR2E1 Q9Y466 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1790721 0.86 TUBB1 (0.50) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL8413308 0.80 ADRB2 (0.55) ADRB2ALDH1A1MEN1CYP1A2CYP2D6
SCHEMBL273429 0.80 ERN1 (0.52) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL8415652 0.79 ADRB2 (0.57) ADRB2ALDH1A1MEN1CYP1A2CYP2D6
SCHEMBL15728130 0.79 TUBB1 (0.61) ALDH1A1SMN1; SMN2KDM4ERAB9ATDP1
SCHEMBL8415057 0.79 KDM4E (0.62) ADRB2KDM4E
SCHEMBL5885093 0.77 TUBB1 (0.59) ALDH1A1SMN1; SMN2KDM4ERAB9A
SCHEMBL27500190 0.77 KDM4E (0.58) ALDH1A1CYP1A2SMN1; SMN2KDM4ERAB9A
Hydrochloric Acid SCHEMBL8416654 0.76 ADRB2 (0.53) ADRB2ALDH1A1MEN1CYP1A2CYP2D6
SCHEMBL4064858 0.75 ALDH1A1 (0.51) ALDH1A1MEN1KMT2ASMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866611-A PHENOXYPROPYLAMINE INHIBITORS OF SQUALENE SYNTHESE, USEFUL IN TREATING DISEASES IN WHICH A LOWERING OF CHOLESTEROL IS DESIRABLE. ZENECA LIMITED (GB) 1999-02-02 US disclosed
EP-0589018-A1 AMINES AS INHIBITORS OF SQUALENE SYNTHASE ZENECA LIMITED (GB) 1994-03-30 EP disclosed
WO-1993020807-A1 AMINES AS INHIBITORS OF SQUALENE SYNTHASE ZENECA LIMITED (GB) 1993-10-28 WO disclosed