SCHEMBL8414903

SCHEMBL8414903

CCOC(=O)Oc1cc2cc(Cl)ccc2nc1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 3/20 0.44
HPGD P15428 1/20 0.44
PTPN1 P18031 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RXFP1 Q9HBX9 1/20 0.41
ALOX15 P16050 1/20 0.40
ADORA2A P29274 1/20 0.40
CA2 P00918 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
SIRT3 Q9NTG7 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9677441 0.89 PTPN1 (0.41) TSHRALDH1A1KDM4EHPGDPTPN1
SCHEMBL6824035 0.79 TSHR (0.71) TSHRALDH1A1KDM4EHPGDL3MBTL1
SCHEMBL4089116 0.76 SMN1; SMN2 (0.52) TSHRALDH1A1KDM4EHPGDMAPT
SCHEMBL24453339 0.74 PPARG (0.48) TSHRHPGDSMN1; SMN2ALOX15MEN1
SCHEMBL2314666 0.73 TSHR (0.56) TSHRALDH1A1KDM4EHPGDMAPT
SCHEMBL18050527 0.72 MAPK1 (0.48) TSHRKDM4EMAPTLMNAHTT
SCHEMBL10665205 0.72 TSHR (0.58) TSHRALDH1A1KDM4EHPGDMAPT
SCHEMBL17375002 0.71 ALDH1A1 (0.42) TSHRALDH1A1KDM4EHPGDL3MBTL1
SCHEMBL13651187 0.71 KDM4E (0.45) ALDH1A1KDM4EL3MBTL1LMNASMN1; SMN2
SCHEMBL15124569 0.71 ADORA2A (0.49) TSHRALDH1A1KDM4EHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0682017-B1 Substituted bicycle heteroaroylguanidines, their preparation and their application in medicaments and diagnostic agents HOECHST AG (DE) 1999-08-11 EP disclosed
EP-0682017-A1 Substituted bicycle heteroaroylguanidines, their preparation and their application in medicaments and diagnostic agents HOECHST AKTIENGESELLSCHAFT (DE) 1995-11-15 EP disclosed