SCHEMBL8416489

SCHEMBL8416489

COc1cc(O)c(C(=O)NC(=O)[C@@H]2CCCN2)c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTR2C P28335 5/20 0.39
HTR2B P41595 4/20 0.39
HTR2A P28223 2/20 0.38
AAK1 Q2M2I8 1/20 0.38
GHSR Q92847 4/20 0.38
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
DPP4 P27487 1/20 0.36
SUV39H2 Q9H5I1 1/20 0.36
CTSC P53634 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8419532 0.81 PLK1 (0.53) KDM4ECYP3A4CYP2D6CYP1A2CYP2C19
SCHEMBL11121066 0.80 KDM4E (0.47) KDM4ECYP3A4CYP2D6CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL7267342 0.80 KDM4E (0.47) KDM4ECYP3A4CYP2D6CYP1A2CYP2C19
SCHEMBL13570608 0.78 TDP1 (0.49) KDM4ECYP3A4CYP2D6CYP1A2CYP2C19
SCHEMBL7517030 0.74 CDC25B (0.46) KDM4ECYP3A4CYP2D6CYP1A2CYP2C19
SCHEMBL8419535 0.74 KDM4E (0.52) KDM4ECYP3A4CYP2D6CYP1A2CYP2C19
SCHEMBL4614497 0.73 AAK1 (0.50) KDM4ECYP3A4CYP2D6CYP1A2CYP2C19
SCHEMBL9643299 0.73 AAK1 (0.50) KDM4ECYP3A4CYP2D6CYP1A2CYP2C19
SCHEMBL13570366 0.71 GPR6 (0.49) TSHR
SCHEMBL8397188 0.70 CTSC (0.49) CYP3A4CYP2D6CYP1A2CYP2C19HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0791071-B1 ASSAY FOR PROLINE IMINOPEPTIDASE AND OTHER HYDROLYTIC ACTIVITIES LITMUS CONCEPTS INC (US) 1999-09-15 EP disclosed
EP-0791071-A1 ASSAY FOR PROLINE IMINOPEPTIDASE AND OTHER HYDROLYTIC ACTIVITIES LITMUS CONCEPTS, INC. (US) 1997-08-27 EP disclosed
US-5571684-A SOLID PHASE CONJUGATE LITMUS CONCEPTS, INC. (US) 1996-11-05 US disclosed
WO-1996015255-A2 ASSAY FOR PROLINE IMINOPEPTIDASE AND OTHER HYDROLYTIC ACTIVITIES LITMUS CONCEPTS, INC. (US) 1996-05-23 WO disclosed