SCHEMBL8417660

SCHEMBL8417660

COCCOC(=O)C=Cc1ccc(O)cc1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B10 O60218 8/20 0.58
AKR1B1 P15121 8/20 0.58
ALOX5 P09917 1/20 0.51
ESR1 P03372 2/20 0.48
ALDH1A1 P00352 2/20 0.48
MAPT P10636 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
CYP2C19 P33261 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MET P08581 2/20 0.46
CA12 O43570 3/20 0.46
CA1 P00915 3/20 0.46
CA7 P43166 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8417663 1.00 AKR1B10 (0.58) AKR1B10AKR1B1ALOX5ESR1ALDH1A1
SCHEMBL15960946 0.85 ESR1 (0.62) AKR1B10AKR1B1ESR1ALDH1A1MAPT
SCHEMBL9820613 0.84 APP (0.57) AKR1B10AKR1B1ESR1CA12CA1
SCHEMBL18993841 0.83 AKR1B10 (0.49) AKR1B10AKR1B1ALOX5ESR1ALDH1A1
SCHEMBL9820607 0.77 TYR (0.53) AKR1B10AKR1B1ESR1ALDH1A1MAPT
SCHEMBL20888287 0.77 AKR1B10 (0.71) AKR1B10AKR1B1ALOX5ESR1ALDH1A1
SCHEMBL8417664 0.76 ALDH1A1 (0.49) AKR1B10AKR1B1ESR1ALDH1A1MAPT
SCHEMBL10021706 0.75 CAPN1 (0.50) ALDH1A1MAPTMEN1CYP1A2CYP2C9
SCHEMBL8148901 0.75 ESR1 (0.45) AKR1B10AKR1B1ALOX5ESR1ALDH1A1
SCHEMBL8420014 0.75 AKR1B10 (0.47) AKR1B10AKR1B1ALOX5METCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919793-A QUINUCLIDINE DERIVATIVES, SQUALENE SYNTHETASE INHIBITORS, ANTICHOLESTEROL AGENTS ZENECA LIMITED (GB) 1999-07-06 US disclosed
EP-0696284-A1 HETEROCYCLIC DERIVATIVES ZENECA LIMITED (GB) 1996-02-14 EP disclosed
WO-1994025459-A1 HETEROCYCLIC DERIVATIVES ZENECA LIMITED (GB) 1994-11-10 WO disclosed