SCHEMBL8417751

SCHEMBL8417751

COCCOCCc1ccc(Br)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.45
HTR2A P28223 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
KDM4E B2RXH2 1/20 0.45
GLA P06280 1/20 0.45
MAPT P10636 2/20 0.40
POLB P06746 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
ALDH1A1 P00352 1/20 0.40
IDO1 P14902 2/20 0.39
MAOB P27338 2/20 0.37
MAOA P21397 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
KCNH2 Q12809 1/20 0.37
THRB P10828 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21382605 0.92 L3MBTL1 (0.42) TAAR1HTR2AL3MBTL1KDM4EGLA
SCHEMBL517859 0.89 TAAR1 (0.50) TAAR1HTR2AL3MBTL1KDM4EGLA
SCHEMBL2515837 0.89 TAAR1 (0.54) TAAR1HTR2APOLBCTDSP1IDO1
SCHEMBL2172552 0.86 TAAR1 (0.44) TAAR1HTR2AL3MBTL1KDM4EGLA
SCHEMBL18218371 0.85 L3MBTL1 (0.46) TAAR1HTR2AL3MBTL1KDM4EGLA
SCHEMBL19792648 0.84 RAD52 (0.39) TAAR1L3MBTL1KDM4EGLAMAPT
SCHEMBL26987687 0.83 TAAR1 (0.50) TAAR1HTR2AL3MBTL1KDM4EGLA
SCHEMBL8447026 0.83 KCNH2 (0.51) TAAR1MAPTALDH1A1IDO1MEN1
SCHEMBL1680408 0.83 TAAR1 (0.45) TAAR1HTR2AL3MBTL1POLBCTDSP1
SCHEMBL15602862 0.83 IDO1 (0.48) L3MBTL1KDM4EGLAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919793-A QUINUCLIDINE DERIVATIVES, SQUALENE SYNTHETASE INHIBITORS, ANTICHOLESTEROL AGENTS ZENECA LIMITED (GB) 1999-07-06 US disclosed
CN-1121718-A Heterocyclic derivatives ZENECA LTD (GB) 1996-05-01 CN disclosed
EP-0696284-A1 HETEROCYCLIC DERIVATIVES ZENECA LIMITED (GB) 1996-02-14 EP disclosed
WO-1994025459-A1 HETEROCYCLIC DERIVATIVES ZENECA LIMITED (GB) 1994-11-10 WO disclosed