SCHEMBL8420064

SCHEMBL8420064

NS(=O)(=O)c1ccc(-n2nc(OC(=O)c3ccccc3)cc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.62
CHRNA7 P36544 6/20 0.60
MAPK9 P45984 1/20 0.59
PTGS2 P35354 8/20 0.58
PTGS1 P23219 4/20 0.58
PDPK1 O15530 1/20 0.55
CA9 Q16790 2/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8420104 0.90 PTGS2 (0.54) SMN1; SMN2CHRNA7MAPK9PTGS2PTGS1
SCHEMBL8423935 0.82 CHRNA7 (0.57) SMN1; SMN2CHRNA7MAPK9PTGS2PTGS1
SCHEMBL28190691 0.80 KMT2A (0.62) PTGS1
SCHEMBL27436439 0.78 PTGS2 (0.63) SMN1; SMN2CHRNA7PTGS2PTGS1PDPK1
SCHEMBL8119257 0.78 PTGS2 (0.67) SMN1; SMN2CHRNA7MAPK9PTGS2PTGS1
SCHEMBL212707 0.78 PTGS2 (0.80) CHRNA7MAPK9PTGS2PTGS1PDPK1
SCHEMBL3873219 0.78 CHRNA7 (0.80) SMN1; SMN2CHRNA7MAPK9PTGS2
SCHEMBL8119702 0.78 PTGS2 (0.74) SMN1; SMN2CHRNA7PTGS2PTGS1
SCHEMBL8126719 0.78 PTGS2 (0.74) SMN1; SMN2CHRNA7PTGS2PTGS1
SCHEMBL7156590 0.78 MALT1 (0.58) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed