SCHEMBL8423935

SCHEMBL8423935

NS(=O)(=O)c1ccc(-n2nc(-c3ccc(Cl)cc3)cc2OC(=O)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.57
PTGS2 P35354 9/20 0.54
PTGS1 P23219 4/20 0.54
CA1 P00915 3/20 0.52
CA2 P00918 3/20 0.52
CA9 Q16790 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MMP2 P08253 1/20 0.50
CYP2C9 P11712 1/20 0.50
MAPK9 P45984 1/20 0.49
CA4 P22748 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8423812 0.90 PTGS2 (0.54) CHRNA7PTGS2PTGS1SMN1; SMN2
SCHEMBL8420064 0.82 SMN1; SMN2 (0.62) CHRNA7PTGS2PTGS1CA1CA2
SCHEMBL8733986 0.79 PTGS2 (0.60) PTGS2PTGS1CA1CA2CA9
SCHEMBL212707 0.78 PTGS2 (0.80) CHRNA7PTGS2PTGS1MMP2CYP2C9
SCHEMBL8692916 0.78 PTGS2 (0.60) PTGS2PTGS1CA1CA2CA9
SCHEMBL8120201 0.78 PTGS2 (0.66) CHRNA7PTGS2PTGS1SMN1; SMN2MMP2
SCHEMBL8119702 0.78 PTGS2 (0.74) CHRNA7PTGS2PTGS1SMN1; SMN2CYP2C9
SCHEMBL8126719 0.78 PTGS2 (0.74) CHRNA7PTGS2PTGS1SMN1; SMN2CYP2C9
SCHEMBL8126788 0.77 PTGS2 (0.74) CHRNA7PTGS2PTGS1SMN1; SMN2CYP2C9
SCHEMBL8122672 0.77 PTGS2 (0.74) CHRNA7PTGS2PTGS1SMN1; SMN2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed