SCHEMBL8422280

SCHEMBL8422280

N#Cc1c(-c2ccc(Cl)cc2)nn(NS(=O)(=O)c2ccccc2)c1-c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 4/20 0.41
ALOX5 P09917 4/20 0.41
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
MALT1 Q9UDY8 2/20 0.39
NPSR1 Q6W5P4 2/20 0.38
KDM1A O60341 1/20 0.38
LMNA P02545 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
HPGD P15428 1/20 0.37
GRM5 P41594 2/20 0.37
CDC25A P30304 1/20 0.37
CDC25B P30305 1/20 0.37
NAT1 P18440 1/20 0.37
AURKA O14965 1/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8421920 0.84 PTGES (0.44) PTGESALOX5MALT1NPSR1KDM1A
SCHEMBL8689212 0.82 PTGS1 (0.51) PTGESALOX5MALT1NPSR1KDM1A
SCHEMBL8423988 0.82 PTGES (0.43) PTGESALOX5MALT1NPSR1KDM1A
SCHEMBL8424009 0.82 PTGES (0.43) PTGESALOX5MALT1NPSR1KDM1A
SCHEMBL8424177 0.82 PTGES (0.43) PTGESALOX5MALT1NPSR1KDM1A
SCHEMBL8423891 0.82 ALDH1A1 (0.43) PTGESALOX5MALT1NPSR1KDM1A
SCHEMBL8422206 0.81 PTGES (0.42) PTGESALOX5MALT1NPSR1KDM1A
SCHEMBL8421700 0.79 PTGES (0.43) PTGESALOX5MALT1NPSR1KDM1A
SCHEMBL8422345 0.79 PTGES (0.41) PTGESALOX5MALT1NPSR1KDM1A
SCHEMBL8421861 0.79 PTGES (0.41) PTGESALOX5MALT1NPSR1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed