SCHEMBL8422369

SCHEMBL8422369

CS(=O)(=O)c1ccc(-n2nc(-c3ccc(Cl)cc3Cl)cc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.70
PTGS1 P23219 4/20 0.55
ALOX5 P09917 1/20 0.50
CHRNA7 P36544 1/20 0.49
MALT1 Q9UDY8 1/20 0.49
CYP2C9 P11712 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8421613 0.91 PTGS2 (0.70) PTGS2PTGS1ALOX5CHRNA7MALT1
SCHEMBL8424001 0.91 PTGS2 (0.70) PTGS2PTGS1CHRNA7
SCHEMBL8423791 0.90 PTGS2 (0.69) PTGS2PTGS1ALOX5CHRNA7CYP2C9
SCHEMBL8111892 0.88 PTGS2 (0.70) PTGS2PTGS1CHRNA7CYP2C9
SCHEMBL8420804 0.88 PTGS2 (0.88) PTGS2PTGS1ALOX5MALT1CYP2C9
SCHEMBL8420754 0.85 PTGS2 (0.66) PTGS2PTGS1ALOX5CHRNA7CYP2C9
SCHEMBL8422267 0.85 PTGS2 (0.75) PTGS2PTGS1ALOX5CHRNA7MALT1
SCHEMBL8422328 0.84 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL8420090 0.84 PTGS2 (0.78) PTGS2PTGS1ALOX5CHRNA7MALT1
SCHEMBL8423720 0.84 PTGS2 (0.74) PTGS2PTGS1CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed
US-5434178-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G.D. SEARLE & CO. (US) 1995-07-18 US disclosed