SCHEMBL8423646

SCHEMBL8423646

C=C1CCO[C@@]12CC[C@H]1[C@@H]3CCC4=C/C(=N/O)CC[C@@H]4[C@H]3CC[C@@]12C

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 4/20 0.64
PDK2 Q15119 4/20 0.64
PDK3 Q15120 4/20 0.64
PDK4 Q16654 4/20 0.64
NR1I2 O75469 2/20 0.51
PGR P06401 5/20 0.47
NR3C1 P04150 3/20 0.46
SLC6A4 P31645 2/20 0.46
ADORA3 P0DMS8 2/20 0.46
SLC6A2 P23975 2/20 0.46
AGTR1 P30556 1/20 0.46
DRD3 P35462 1/20 0.46
SLC6A3 Q01959 1/20 0.46
PDE4D Q08499 1/20 0.46
CYP3A4 P08684 3/20 0.45
ABCB11 O95342 3/20 0.45
LMNA P02545 2/20 0.45
CYP2C19 P33261 2/20 0.45
TSHR P16473 1/20 0.45
HIF1A Q16665 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8423647 1.00 PDK1 (0.64) PDK1PDK2PDK3PDK4NR1I2
SCHEMBL8423021 0.84 PGR (0.62) PGRNR3C1SLC6A4ADORA3SLC6A2
SCHEMBL9541216 0.82 PDK1 (0.74) PDK1PDK2PDK3PDK4NR1I2
SCHEMBL8424854 0.80 PGR (0.42) PDK1PDK2PDK3PDK4PGR
SCHEMBL8426916 0.80 PGR (0.42) PDK1PDK2PDK3PDK4PGR
SCHEMBL8423587 0.78 PGR (0.60) PGRNR3C1SLC6A4ADORA3SLC6A2
SCHEMBL5172677 0.78 PDK1 (1.00) PDK1PDK2PDK3PDK4NR1I2
SCHEMBL29653691 0.78 PDK1 (1.00) PDK1PDK2PDK3PDK4NR1I2
SCHEMBL13013574 0.78 AR (0.74) PDK1PDK2PDK3PDK4NR1I2
SCHEMBL8424688 0.75 PGR (0.62) PGRNR3C1SLC6A4ADORA3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582338-B1 17-Spiromethylene steroids AKZO NOBEL NV (NL) 1999-10-20 EP disclosed
US-5854235-A 17-spiromethylene steroids AKZO NOBEL N.V. (NL) 1998-12-29 US disclosed
US-5712264-A 17-spiromethylene steroids AKZO NOBEL N.V. (NL) 1998-01-27 US disclosed
EP-0582338-A2 17-Spiromethylene steroids Akzo Nobel N.V. (NL) 1994-02-09 EP disclosed