SCHEMBL8423930

SCHEMBL8423930

CC(C)c1ccccc1NC(=N)Nc1ccc2cccc3c2c1C=C3

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.39
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
AKR1C3 P42330 1/20 0.37
RECQL P46063 1/20 0.36
KMT2A Q03164 1/20 0.35
MAPT P10636 2/20 0.34
LPAR1 Q92633 3/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
GAA P10253 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6155378 0.85 ALDH1A1 (0.35) MAPTCYP1A2CYP3A4
Bromide SCHEMBL6154601 0.84 ALDH1A1 (0.34) MAPTCYP1A2CYP3A4
SCHEMBL6156250 0.82 GAA (0.43) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8424539 0.81 SIGMAR1 (0.41) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6717468 0.80 GRIN2D (0.40) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6719186 0.80 MAPT (0.39) RECQLKMT2AMAPTGAA
SCHEMBL6719777 0.80 RAB9A (0.38) SIGMAR1KMT2AMAPTCYP1A2GAA
SCHEMBL6724277 0.79 KDM4E (0.45) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6719907 0.78 KDM4E (0.39) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6155354 0.78 SCN2A (0.41) KMT2AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0584088-B1 SUBSTITUTED GUANIDINES AND DERIVATIVES THEREOF AS MODULATORS OF NEUROTRANSMITTER RELEASE AND NOVEL METHODOLOGY FOR IDENTIFYING NEUROTRANSMITTER RELEASE BLOCKERS CAMBRIDGE NEUROSCIENCE RES (US) 1999-10-27 EP claimed