SCHEMBL8423964

SCHEMBL8423964

N#Cc1cccc(CN2CC[C@@H](c3cc(S([NH])(=O)=O)ccc3-c3ccccc3)C2=O)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.41
DRD3 P35462 2/20 0.41
DRD2 P14416 1/20 0.41
F10 P00742 4/20 0.41
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
THRB P10828 1/20 0.38
CHRM3 P20309 1/20 0.38
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
MMP1 P03956 1/20 0.37
ADAM17 P78536 1/20 0.37
KCNH2 Q12809 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8425503 0.81 DRD4 (0.38) DRD4DRD3DRD2F10ROCK2
SCHEMBL2331634 0.77 F10 (0.56) F10
SCHEMBL8423957 0.77 DRD4 (0.42) DRD4DRD3DRD2F10ROCK2
SCHEMBL2328117 0.76 F10 (0.46) DRD4DRD3DRD2F10ROCK2
SCHEMBL8425655 0.75 F10 (0.46) DRD4DRD3DRD2F10KCNH2
SCHEMBL2325190 0.74 F10 (0.68) F10THRB
SCHEMBL8424704 0.73 F10 (0.46) F10
SCHEMBL2332215 0.73 F10 (0.52) DRD4DRD3F10
SCHEMBL12009728 0.69 SIRT2 (0.46) DRD4DRD3DRD2ROCK2ROCK1
SCHEMBL7482530 0.69 SIRT2 (0.48) DRD4DRD3DRD2ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958918-A Substituted (sulfinic acid, sulfonic acid, sulfonylamino or sulfinylamino) N- (aminominomethyl)phenylalkyl!-azaheterocyclylamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. 1999-09-28 US disclosed