SCHEMBL8428161

SCHEMBL8428161

CC1=NN(c2ccc(S(=O)(=O)N3CCN(C)CC3)cc2)C(=O)C1.CCOC(=O)CC(C)=O

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.51
ALDH1A1 P00352 3/20 0.46
LMNA P02545 3/20 0.46
TSHR P16473 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
POLB P06746 1/20 0.43
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8428115 0.90 MAPK1 (0.54) CYP2C9ALDH1A1LMNATSHRPOLB
SCHEMBL6948645 0.85 KMT2A (0.54) ALDH1A1LMNATSHRPOLBATM
SCHEMBL8428070 0.84 CA1 (0.54) ALDH1A1LMNATSHRPOLB
SCHEMBL8428126 0.82 ALDH1A1 (0.43) ALDH1A1LMNATSHRPOLB
SCHEMBL8423248 0.82 APP (0.43) ALDH1A1LMNATSHR
SCHEMBL8427533 0.80 MAPT (0.65) ALDH1A1LMNATSHRPOLB
SCHEMBL8425552 0.79 POLB (0.55) ALDH1A1LMNATSHRPOLB
SCHEMBL6948663 0.73 POLB (0.52) ALDH1A1LMNATSHRPOLB
SCHEMBL9025227 0.72 ALDH1A1 (0.46) CYP2C9ALDH1A1LMNA
SCHEMBL8425824 0.71 KMT2A (0.49) ALDH1A1TSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5869516-A 4-(arylaminomethylene)-2,4-dihydro-3-pyrazolones MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-02-09 US disclosed